SCHEMBL4959110

SCHEMBL4959110

CS(=O)(=O)c1ccc(-c2[nH]nc(CO)c2Cc2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.48
PTGS1 P23219 5/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4958867 0.84 PTGS2 (0.46) PTGS2PTGS1
SCHEMBL6590005 0.83 PTGS2 (0.43) PTGS2PTGS1
SCHEMBL4958540 0.82 PTGS2 (0.44) PTGS2PTGS1
SCHEMBL6438225 0.82 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL8487155 0.77 PTGS2 (0.52) PTGS2PTGS1
SCHEMBL4958133 0.76 PTGS2 (0.44) PTGS2PTGS1
SCHEMBL6589445 0.75 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL18302450 0.73 HCAR2 (0.45)
SCHEMBL6438544 0.73 PTGS2 (0.50) PTGS2PTGS1
SCHEMBL3868483 0.72 MAPK1 (0.36) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1542972-A4 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2008-01-23 EP claimed
EP-1542972-A2 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-22 EP claimed
WO-2004010945-A2 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-02-05 WO claimed
EP-1542972-A4 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2008-01-23 EP disclosed
EP-1542972-A2 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-22 EP disclosed
WO-2004010945-A2 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-02-05 WO disclosed