SCHEMBL4966564

SCHEMBL4966564

NC(=O)Oc1ccc2c(c1)CCc1cc(CNCCCN3CCOCC3)ccc1O2

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C19 P33261 2/20 0.44
CYP3A4 P08684 1/20 0.44
ALDH1A1 P00352 2/20 0.44
PARP1 P09874 2/20 0.42
MAPT P10636 1/20 0.41
BCHE P06276 1/20 0.40
HTT P42858 1/20 0.40
POLB P06746 1/20 0.39
KCNH2 Q12809 1/20 0.39
CACNA1H O95180 1/20 0.39
CACNA1B Q00975 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4968054 0.94 PARP1 (0.43) MEN1KMT2ACYP2D6CYP2C19CYP3A4
SCHEMBL4966170 0.86 KDM4E (0.48) MEN1KMT2ACYP2D6CYP2C19CYP3A4
SCHEMBL4965202 0.84 KDM4E (0.45) MEN1KMT2ACYP2D6CYP2C19CYP3A4
SCHEMBL4965638 0.82 OPRM1 (0.41) CYP2D6CYP2C19
SCHEMBL4965138 0.82 MCHR1 (0.43) MEN1KMT2AALDH1A1POLB
SCHEMBL4963457 0.82 SLC2A1 (0.42) CYP2D6CYP2C19
SCHEMBL4968023 0.81 OPRM1 (0.46) MAPTPOLBKCNH2
SCHEMBL4965633 0.81 OPRM1 (0.45) MEN1KMT2ACYP2D6CYP2C19CYP3A4
SCHEMBL4966629 0.81 SLC2A1 (0.37) MEN1KMT2ACYP2D6CYP2C19CYP3A4
SCHEMBL4967478 0.80 KDM4E (0.49) MEN1KMT2AALDH1A1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730140-B1 OPIOID RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-06-25 EP claimed