SCHEMBL5148555

SCHEMBL5148555

CC[N+](C)(CC)C1Cc2cc(C)cc(-c3ccc(OC)cc3)c2O1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.37
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
MAOB P27338 4/20 0.33
F2RL3 Q96RI0 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
ATM Q13315 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
SYK P43405 1/20 0.32
ABL1 P00519 1/20 0.32
ABCB1 P08183 1/20 0.32
BCR P11274 1/20 0.32
ACLY P53396 1/20 0.31
GSK3B P49841 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4823949 0.87 AQP1 (0.31) MAPTTDP1
SCHEMBL4596468 0.80 ALDH1A1 (0.42) DRD2ALDH1A1MAPTMAOBF2RL3
SCHEMBL4596465 0.79 ALDH1A1 (0.37) DRD2ALDH1A1MAPTMAOBF2RL3
SCHEMBL4222368 0.78 PRKAB2 (0.51) DRD2ALDH1A1MAPTMAOBF2RL3
SCHEMBL5148557 0.77 DRD2 (0.38) DRD2ALDH1A1MAPTMAOBF2RL3
SCHEMBL4226625 0.76 PRKAB2 (0.42) DRD2ALDH1A1MAPTMAOBF2RL3
SCHEMBL4226616 0.76 AQP1 (0.45) DRD2ALDH1A1MAPTMAOBF2RL3
SCHEMBL4970746 0.75 AQP1 (0.46) ALDH1A1F2RL3MAPK1HSD17B10
SCHEMBL4836377 0.75 AQP1 (0.36) ALDH1A1MAPTMAPK1HTTTDP1
SCHEMBL6047897 0.72 GSK3B (0.38) DRD2ALDH1A1MAPTMAOBSYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1871354-A1 TREATMENT OF PAIN Wyeth (US) 2008-01-02 EP disclosed
WO-2006116171-A1 TREATMENT OF PAIN WYETH (US) 2006-11-02 WO disclosed