SCHEMBL4972736

SCHEMBL4972736

CCOC(=O)c1ccc(C[C@@H]2CN(Cc3ccccc3)CCN2C(=O)O)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.57
CA1 P00915 2/20 0.55
CA2 P00918 2/20 0.55
CA4 P22748 2/20 0.55
CA9 Q16790 2/20 0.55
MAPK1 P28482 1/20 0.54
PRMT1 Q99873 1/20 0.51
ALDH1A1 P00352 1/20 0.51
TSHR P16473 1/20 0.51
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
NPC1 O15118 1/20 0.48
TNF P01375 1/20 0.48
RAB9A P51151 1/20 0.48
NOD2 Q9HC29 1/20 0.48
NOD1 Q9Y239 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
DPP4 P27487 1/20 0.46
DPP7 Q9UHL4 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3494268 0.88 LMNA (0.52) LMNACA1CA2CA4CA9
SCHEMBL3494525 0.85 CA1 (0.63) CA1CA2CA4CA9DPP4
SCHEMBL3496196 0.83 RAB9A (0.44) CA1CA2CA4CA9MAPK1
SCHEMBL13341229 0.82 L3MBTL1 (0.54) LMNACA1CA2CA4CA9
SCHEMBL3495202 0.82 CA2 (0.57) CA1CA2CA4CA9DPP4
SCHEMBL3495256 0.81 CA1 (0.47) LMNACA1CA2CA4CA9
SCHEMBL4287508 0.81 CA1 (0.56) LMNACA1CA2CA4CA9
SCHEMBL1714109 0.79 AGTR2 (0.51) CA1CA2CA4CA9ALDH1A1
SCHEMBL3494272 0.79 OPRD1 (0.45) LMNACA1CA2CA4CA9
SCHEMBL3492288 0.79 CA1 (0.54) CA1CA2CA4CA9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1984355-A2 CYCLIC AMINE COMPOUND AND USE THEREOF FOR THE PROPHYLAXIS OR TREATMENT OF HYPERTENSION Takeda Pharmaceutical Company Limited (JP) 2008-10-29 EP disclosed
WO-2007094513-A2 CYCLIC AMINE COMPOUND AND USE THEREOF FOR THE PROPHYLAXIS OR TREATMENT OF HYPERTENSION TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-08-23 WO disclosed