SCHEMBL4974117

SCHEMBL4974117

CC(C)(C)N1CCC[C@@H]([C@@H](OCCN)c2ccc(F)c(Cl)c2)C1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 4/20 0.40
SLC6A4 P31645 4/20 0.40
SLC6A3 Q01959 3/20 0.40
KCNH2 Q12809 1/20 0.36
REN P00797 10/20 0.36
DPP4 P27487 1/20 0.36
DPP8 Q6V1X1 1/20 0.36
DPP9 Q86TI2 1/20 0.36
DPP7 Q9UHL4 1/20 0.36
CHRNB1 P11230 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNB3 Q05901 1/20 0.33
CYP3A4 P08684 2/20 0.33
TACR1 P25103 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4973673 0.87 REN (0.47) SLC6A2SLC6A4SLC6A3RENCYP3A4
SCHEMBL3968254 0.87 REN (0.47) SLC6A2SLC6A4SLC6A3RENCYP3A4
SCHEMBL4971174 0.86 SLC6A3 (0.36) SLC6A2SLC6A4SLC6A3KCNH2REN
SCHEMBL4974711 0.86 REN (0.43) RENCYP3A4
SCHEMBL4973483 0.84 REN (0.53) RENCYP3A4
SCHEMBL2326128 0.82 REN (0.44) RENDPP4DPP8DPP9DPP7
SCHEMBL2326131 0.82 REN (0.44) RENDPP4DPP8DPP9DPP7
SCHEMBL2326129 0.82 REN (0.44) RENDPP4DPP8DPP9DPP7
SCHEMBL4972006 0.81 REN (0.41) RENCYP3A4
SCHEMBL4969812 0.81 REN (0.45) REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966139-A1 ASPARTIC PROTEASE INHIBITORS Vitae Pharmaceuticals, Inc. (US) 2008-09-10 EP disclosed
WO-2007070201-A1 ASPARTIC PROTEASE INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2007-06-21 WO disclosed