SCHEMBL499193

SCHEMBL499193

CC(C)N(CCC(O)c1cccc(Cl)c1)C(=O)OC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 12/20 0.39
ADRB1 P08588 10/20 0.39
ADRB2 P07550 10/20 0.39
CYP2D6 P10635 2/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
BACE1 P56817 1/20 0.38
GLA P06280 1/20 0.38
SLC2A1 P11166 2/20 0.38
CYP3A4 P08684 1/20 0.37
HIF1A Q16665 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL499535 0.87 RIPK1 (0.38) ADRB3ADRB1ADRB2CYP2D6ADRA1D
SCHEMBL4755330 0.84 ADRB3 (0.45) ADRB3ADRB1ADRB2CYP2D6ADRA1D
SCHEMBL27656228 0.82 BACE1 (0.43) ADRB3ADRB1ADRB2CYP2D6ADRA1D
SCHEMBL499034 0.80 LMNA (0.38) CYP1A2CYP2C19
SCHEMBL9316827 0.76 BACE1 (0.46) ADRB3ADRB1ADRB2CYP2D6ADRA1D
SCHEMBL27693712 0.76 BACE1 (0.46) ADRB3ADRB1ADRB2CYP2D6ADRA1D
SCHEMBL8770902 0.76 L3MBTL1 (0.43) ADRB3ADRB1ADRB2CYP2D6ADRA1D
SCHEMBL10318009 0.76 KDM4E (0.46) CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL7120069 0.76 BACE1 (0.43) ADRB3ADRB1ADRB2CYP2D6ADRA1D
SCHEMBL7120076 0.76 BACE1 (0.43) ADRB3ADRB1ADRB2CYP2D6ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106221-B2 Renin inhibitors VITAE PHARMACEUTICALS, INC. (US) 2012-01-31 US disclosed
US-8106221-B2 Renin inhibitors VITAE PHARMACEUTICALS, INC. (US) 2012-01-31 US disclosed
US-20100144825-A1 Renin Inhibitors VITAE PHARMACEUTICALS, INC. 2010-06-10 US disclosed
US-20100144825-A1 Renin Inhibitors VITAE PHARMACEUTICALS, INC. 2010-06-10 US disclosed
WO-2008156816-A2 RENIN INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2008-12-24 WO disclosed
WO-2008156816-A2 RENIN INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2008-12-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100144825-A1 Renin Inhibitors ACE, REN, DNPEP ADRB3 1089/4885ADRB1 1050/4885ADRB2 1697/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.