SCHEMBL5011684

SCHEMBL5011684

COc1ccc(NC(=O)ON2N(Cc3ccccc3)C(=O)OC23CCCCC3)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.47
FAAH O00519 2/20 0.47
TRPV1 Q8NER1 1/20 0.47
ALDH1A1 P00352 3/20 0.43
MAPT P10636 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
RAB9A P51151 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
EP300 Q09472 2/20 0.43
NCOA1 Q15788 1/20 0.43
NCOA3 Q9Y6Q9 1/20 0.43
CNR2 P34972 1/20 0.42
OPRD1 P41143 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
AKR1B1 P15121 1/20 0.42
TP53 P04637 1/20 0.41
HTT P42858 2/20 0.41
CACNA1G O43497 1/20 0.41
CACNA1H O95180 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5013591 0.88 TSHR (0.47) LMNAFAAHTRPV1ALDH1A1MAPT
SCHEMBL5011711 0.80 MAPT (0.46) LMNAFAAHTRPV1ALDH1A1MAPT
SCHEMBL5015097 0.76 ALDH1A1 (0.42) LMNAFAAHTRPV1ALDH1A1MAPT
SCHEMBL4257512 0.74 LMNA (0.48) LMNAFAAHTRPV1ALDH1A1MAPT
SCHEMBL4032463 0.66 CCR3 (0.47) LMNAFAAHALDH1A1MAPTSMN1; SMN2
SCHEMBL1223807 0.65 RAB9A (0.67) LMNAALDH1A1MAPTSMN1; SMN2RAB9A
SCHEMBL9818694 0.65 CNR1 (0.62) ALDH1A1MAPTRAB9AL3MBTL1NPC1
SCHEMBL16383892 0.65 KDM4E (0.74) LMNAFAAHTRPV1ALDH1A1MAPT
SCHEMBL12478886 0.64 ACHE (0.60) LMNAALDH1A1MAPTSMN1; SMN2HTT
SCHEMBL5011708 0.64 CYP1A2 (0.45) LMNAALDH1A1MAPTSMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910381-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-04-16 EP disclosed
WO-2007000325-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-01-04 WO disclosed