SCHEMBL5013364

SCHEMBL5013364

[O]c1cc2ncsc2cc1N1CCN(Cc2ccc(OC(F)(F)F)cc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.50
ALDH1A1 P00352 1/20 0.47
LSS P48449 1/20 0.42
DRD2 P14416 7/20 0.41
TEAD1 P28347 2/20 0.40
DRD4 P21917 2/20 0.40
SCN9A Q15858 1/20 0.40
NTRK1 P04629 1/20 0.39
NTRK2 Q16620 1/20 0.39
PHGDH O43175 1/20 0.39
GPR6 P46095 1/20 0.38
NAMPT P43490 1/20 0.38
DRD3 P35462 1/20 0.38
HTR1A P08908 1/20 0.38
HTR2A P28223 1/20 0.38
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
BACE1 P56817 1/20 0.38
PPARD Q03181 1/20 0.38
PPARA Q07869 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2088515 0.84 NTRK1 (0.38) NTRK1NTRK2DRD3
SCHEMBL27666102 0.80 TSHR (0.50) TSHRALDH1A1LSSDRD2TEAD1
SCHEMBL5015139 0.73 PPARD (0.43) TSHRALDH1A1LSSDRD2DRD4
SCHEMBL5013349 0.72 KCNN4 (0.46) TSHRALDH1A1DRD2DRD4GPR6
SCHEMBL5543182 0.70 ALDH1A1 (0.62) TSHRALDH1A1LSSDRD2DRD4
SCHEMBL8170370 0.69 ALDH1A1 (0.58) TSHRALDH1A1LSSDRD2DRD4
SCHEMBL5016235 0.68 RAB9A (0.46) ALDH1A1DRD2DRD4DRD3
SCHEMBL5016362 0.67 CASP1 (0.38) ALDH1A1DRD2DRD4DRD3
SCHEMBL2090465 0.67 SCN4A (0.56) TSHRALDH1A1SCN9APHGDHPPARD
SCHEMBL2056209 0.67 RAB9A (0.57) TSHRALDH1A1SCN9APHGDHPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678185-B1 2,3-DIHYDRO-6-NITROIMIDAZO [2,1-B] OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMA CO LTD (JP) 2008-10-08 EP disclosed