SCHEMBL5014328

SCHEMBL5014328

CCCc1[c]cccc1NS(=O)(=O)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 3/20 0.50
ALDH1A1 P00352 4/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
TSHR P16473 2/20 0.47
KMT2A Q03164 1/20 0.47
RECQL P46063 1/20 0.45
AGTR1 P30556 1/20 0.45
GLO1 Q04760 1/20 0.45
PAX8 Q06710 1/20 0.45
SLC40A1 Q9NP59 1/20 0.45
POLB P06746 2/20 0.43
KCNA5 P22460 1/20 0.42
GAA P10253 1/20 0.42
HTT P42858 1/20 0.42
IL1RN P18510 1/20 0.42
KEAP1 Q14145 1/20 0.42
ERAP1 Q9NZ08 1/20 0.42
USP2 O75604 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5012855 0.81 KEAP1 (0.42) TSHRKMT2AGLO1GAAHTT
SCHEMBL10438570 0.78 ALDH1A1 (0.57) METAP2ALDH1A1SMN1; SMN2TSHRKMT2A
SCHEMBL4573379 0.78 ALDH1A1 (0.54) METAP2ALDH1A1SMN1; SMN2TSHRKMT2A
SCHEMBL28800836 0.75 ALDH1A1 (0.50) ALDH1A1SMN1; SMN2TSHRKMT2ARECQL
SCHEMBL28740683 0.74 ALDH1A1 (0.57) METAP2ALDH1A1SMN1; SMN2TSHRKMT2A
SCHEMBL2207251 0.74 METAP2 (0.48) METAP2ALDH1A1SMN1; SMN2TSHRKMT2A
SCHEMBL2207344 0.74 METAP2 (0.48) METAP2ALDH1A1SMN1; SMN2TSHRKMT2A
SCHEMBL8667928 0.74 KDM4E (0.32) ALDH1A1RECQLPOLBUSP2MAPT
SCHEMBL5892150 0.74 IDO1 (0.34) TSHRKMT2ARECQLUSP2
SCHEMBL2067538 0.73 ALDH1A1 (0.68) METAP2ALDH1A1SMN1; SMN2KMT2ARECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888596-A1 SUBSTITUTED SPIRO COMPOUNDS AND THEIR USE FOR PRODUCING PAIN-RELIEF MEDICAMENTS Grünenthal GmbH (DE) 2008-02-20 EP disclosed
WO-2006122770-A1 SUBSTITUTED SPIRO COMPOUNDS AND THEIR USE FOR PRODUCING PAIN-RELIEF MEDICAMENTS Grünenthal GmbH (DE) 2006-11-23 WO disclosed