SCHEMBL5014672

SCHEMBL5014672

C[S+]([O-])c1cccc(-c2ccc(C(C)(C)O)cc2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.39
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36
PGR P06401 1/20 0.35
TNKS O95271 2/20 0.34
PARP1 P09874 2/20 0.34
TNKS2 Q9H2K2 2/20 0.34
DHODH Q02127 1/20 0.34
ASIC1 P78348 1/20 0.34
CYP2C9 P11712 2/20 0.33
HSD17B2 P37059 2/20 0.33
CYP3A4 P08684 1/20 0.33
HSD17B1 P14061 1/20 0.33
MEN1 O00255 1/20 0.33
ESR1 P03372 1/20 0.33
KMT2A Q03164 1/20 0.33
KIF11 P52732 1/20 0.33
KCNH2 Q12809 2/20 0.33
GRM2 Q14416 1/20 0.33
CREBBP Q92793 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20048840 0.79 MAOA (0.41) CYP2C9HSD17B2CYP3A4HSD17B1PTPN1
SCHEMBL547993 0.77 RXRA (0.51) SYKRXRARXRBPGRTNKS
Hydrogen Sulfide SCHEMBL28009272 0.77 MAOA (0.40) PTPN1
SCHEMBL4517154 0.77 CYP2C9 (0.48) SYKRXRARXRBTNKSPARP1
SCHEMBL10802069 0.73 PGR (0.61) SYKPGRTNKSPARP1TNKS2
SCHEMBL4506291 0.72 CYP2C9 (0.56) TNKSPARP1TNKS2CYP2C9CYP3A4
SCHEMBL429422 0.72 CYP2C9 (0.56) TNKSPARP1TNKS2CYP2C9CYP3A4
SCHEMBL21770501 0.72 TAAR1 (0.39) CYP2C9HSD17B2CYP3A4HSD17B1MEN1
SCHEMBL18802754 0.72 KIF11 (0.44) TNKSPARP1TNKS2CYP2C9CYP3A4
SCHEMBL547767 0.72 KIF11 (0.44) TNKSPARP1TNKS2CYP2C9CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893562-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B Merck Frosst Canada Ltd. (CA) 2008-03-05 EP disclosed
WO-2006133559-A1 REVERSIBLE INHIBITORS OF MONOAMINE OXIDASE A AND B MERCK FROSST CANADA LTD. (CA) 2006-12-21 WO disclosed