SCHEMBL5034905

SCHEMBL5034905

O=C(NCCc1c[nH]cn1)Oc1csc(N(C(=O)c2ccc(Cl)cc2Cl)c2ccc(Cl)cc2)n1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.35
TP53 P04637 5/20 0.33
MAPT P10636 3/20 0.33
HPGD P15428 2/20 0.32
PDE5A O76074 1/20 0.31
KMT2A Q03164 1/20 0.31
P2RX7 Q99572 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
THRB P10828 1/20 0.31
LMNA P02545 1/20 0.31
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5038811 0.87 KMT2A (0.39) CYP3A4TP53MAPTHPGDPDE5A
SCHEMBL5039137 0.82 POLB (0.40) CYP3A4MAPTHPGDKMT2ASMN1; SMN2
SCHEMBL5039110 0.81 CYP3A4 (0.42) CYP3A4MAPTPDE5AKMT2ATHRB
SCHEMBL5036060 0.77 CYP3A4 (0.43) CYP3A4MAPTHPGDKMT2ASMN1; SMN2
SCHEMBL5041330 0.75 CYP3A4 (0.44) CYP3A4MAPTKMT2ASMN1; SMN2LMNA
SCHEMBL5035268 0.75 LIPE (0.47) CYP3A4HPGDKMT2ACYP11B1CYP11B2
SCHEMBL5032567 0.75 CYP3A4 (0.49) CYP3A4MAPTKMT2ASMN1; SMN2CYP11B1
SCHEMBL5035238 0.75 LIPE (0.45)
SCHEMBL5035237 0.74 POLB (0.46) CYP3A4TP53MAPTHPGDKMT2A
SCHEMBL5036077 0.73 CYP3A4 (0.42) CYP3A4MAPTKMT2ACYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1694673-B1 THIAZOLE DERIVATES HOFFMANN LA ROCHE (CH) 2008-01-16 EP claimed