SCHEMBL5035268

SCHEMBL5035268

CN1CCN(NC(=O)Oc2csc(N(C(=O)c3ccc(Cl)cc3Cl)c3ccc(Cl)cc3)n2)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LIPE Q05469 4/20 0.47
CNR1 P21554 2/20 0.39
CYP3A4 P08684 1/20 0.37
RAB9A P51151 1/20 0.36
HRH4 Q9H3N8 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CNR2 P34972 1/20 0.35
ALDH1A1 P00352 2/20 0.35
CCNT1 O60563 1/20 0.35
CDK4 P11802 1/20 0.35
CCND1 P24385 1/20 0.35
CDK9 P50750 1/20 0.35
CDK6 Q00534 1/20 0.35
KDM4E B2RXH2 1/20 0.34
HPGD P15428 1/20 0.34
KMT2A Q03164 1/20 0.34
GAA P10253 1/20 0.34
POLB P06746 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5035238 0.91 LIPE (0.45) LIPECNR1CNR2
SCHEMBL14190186 0.85 CNR1 (0.44) LIPECNR1CYP3A4RAB9AHRH4
SCHEMBL5039110 0.82 CYP3A4 (0.42) CYP3A4RAB9ATDP1ALDH1A1KDM4E
SCHEMBL5041330 0.80 CYP3A4 (0.44) CNR1CYP3A4RAB9AALDH1A1KDM4E
SCHEMBL5036060 0.79 CYP3A4 (0.43) CYP3A4RAB9AKDM4EHPGDKMT2A
SCHEMBL5039118 0.78 MCHR1 (0.41) CYP3A4CYP11B1CYP11B2
SCHEMBL5032685 0.78 GABRA2 (0.46) CYP3A4RAB9AHRH4ALDH1A1HPGD
SCHEMBL5039137 0.78 POLB (0.40) LIPECYP3A4RAB9AALDH1A1KDM4E
SCHEMBL5032567 0.77 CYP3A4 (0.49) CNR1CYP3A4RAB9ACNR2ALDH1A1
SCHEMBL5034899 0.77 NLRP3 (0.38) CYP3A4KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1694673-B1 THIAZOLE DERIVATES HOFFMANN LA ROCHE (CH) 2008-01-16 EP claimed