Urea

Urea

SCHEMBL5045628

C1CCN(N2CCCCC2)CC1.NC(N)=O

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.44
ALDH1A1 P00352 5/20 0.43
F2 P00734 1/20 0.41
LMNA P02545 1/20 0.40
OR51E2 Q9H255 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
CA2 P00918 3/20 0.36
CA1 P00915 2/20 0.36
HPGD P15428 2/20 0.36
MMP1 P03956 1/20 0.36
MMP2 P08253 1/20 0.36
MMP3 P08254 1/20 0.36
MMP9 P14780 1/20 0.36
NPC1 O15118 1/20 0.35
MAPT P10636 2/20 0.35
GAA P10253 1/20 0.35
CHKA P35790 1/20 0.35
POLB P06746 1/20 0.35
DPP7 Q9UHL4 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Carbamic Acid SCHEMBL29704037 0.90 ACHE (0.44) L3MBTL1ALDH1A1F2CA2CA1
SCHEMBL3375870 0.88 L3MBTL1 (0.41) L3MBTL1ALDH1A1F2CA2CA1
Carbamic Acid SCHEMBL2830897 0.87 ACHE (0.47) L3MBTL1ALDH1A1F2LMNAOR51E2
SCHEMBL3658220 0.78 MGLL (0.40) ALDH1A1F2CA2CA1POLB
Cycloheptane SCHEMBL1834654 0.78 LMNA (0.67) L3MBTL1ALDH1A1LMNAOR51E2TDP1
Cyclohexane SCHEMBL3125968 0.78 LMNA (0.67) L3MBTL1ALDH1A1LMNAOR51E2TDP1
Cyclohexane SCHEMBL1841235 0.78 LMNA (0.67) L3MBTL1ALDH1A1LMNAOR51E2TDP1
SCHEMBL2457046 0.78 MGLL (0.40) ALDH1A1F2CA2CA1POLB
SCHEMBL42220 0.78 MGLL (0.40) ALDH1A1F2CA2CA1POLB
SCHEMBL6926105 0.78 MGLL (0.40) ALDH1A1F2CA2CA1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1988078-B1 Carboxamide derivatives of pyrrolidine, piperidine and hexahydroazepine for the treatment of thrombosis disorders ORTHO MCNEIL PHARM INC (US) 2012-10-17 EP disclosed
EP-1988078-A1 Carboxamide derivatives of pyrrolidine, piperidine and hexahydroazepine for the treatment of thrombosis disorders Ortho-McNeil Pharmaceutical, Inc. (US) 2008-11-05 EP disclosed
EP-0923555-B1 CARBOXAMIDE DERIVATIVES OF PYRROLIDINE, PIPERIDINE AND HEXAHYDROAZEPINE FOR THE TREATMENT OF THROMBOSIS DISORDERS ORTHO MCNEIL PHARM INC (US) 2005-06-15 EP disclosed
EP-1184374-A1 Carboxamide derivatives of pyrrolidine, piperidine and hexahydroazepine for the treatment of thrombosis disorders ORTHO PHARMACEUTICAL CORPORATION (US) 2002-03-06 EP disclosed
EP-0923555-A1 CARBOXAMIDE DERIVATIVES OF PYRROLIDINE, PIPERIDINE AND HEXAHYDROAZEPINE FOR THE TREATMENT OF THROMBOSIS DISORDERS ORTHO PHARMACEUTICAL CORPORATION (US) 1999-06-23 EP disclosed
WO-1997041102-A1 CARBOXAMIDE DERIVATIVES OF PYRROLIDINE, PIPERIDINE AND HEXAHYDROAZEPINE FOR THE TREATMENT OF THROMBOSIS DISORDERS ORTHO PHARMACEUTICAL CORPORATION (US) 1997-11-06 WO disclosed