SCHEMBL5047653

SCHEMBL5047653

CCCCNC(=O)Oc1cc(-c2csc(-c3cc(OC)cc(OC)c3)n2)n(CC2CCCCC2)c1C

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ATP4A P20648 2/20 0.38
ATP4B P51164 2/20 0.38
CYP1A1 P04798 1/20 0.37
CYP1B1 Q16678 1/20 0.37
CDC25A P30304 1/20 0.35
CDC25B P30305 1/20 0.35
CDC25C P30307 1/20 0.35
DUSP3 P51452 1/20 0.35
MGLL Q99685 2/20 0.34
MAPT P10636 3/20 0.33
TP53 P04637 2/20 0.33
PLA2G2A P14555 1/20 0.33
AVPR1B P47901 2/20 0.32
OXTR P30559 1/20 0.32
AVPR1A P37288 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
ACHE P22303 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5048696 0.93 CDC25A (0.43) ATP4AATP4BCDC25ACDC25BCDC25C
SCHEMBL5044042 0.91 CDC25A (0.42) ATP4AATP4BCDC25ACDC25BCDC25C
SCHEMBL5044496 0.91 ATP4A (0.37) ATP4AATP4BCDC25ACDC25BCDC25C
SCHEMBL5047889 0.89 MGLL (0.36) CDC25ACDC25BCDC25CDUSP3MGLL
SCHEMBL5044102 0.88 MAPT (0.40) ATP4AATP4BMAPTTP53
SCHEMBL5040330 0.88 NTMT1 (0.40) MGLLTP53AVPR1B
SCHEMBL5040235 0.88 HTR2A (0.42) ATP4AATP4BCYP1A1CYP1B1CDC25A
SCHEMBL5133506 0.88 CPT2 (0.40) CDC25ACDC25BCDC25CDUSP3MGLL
SCHEMBL5047187 0.88 HDAC3 (0.36) MGLLACHE
SCHEMBL5039575 0.85 AR (0.43) MGLLMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583762-B1 PYRROLYL-THIAZOLES AND THEIR USE AS CB 1 RECEPTOR INVERSE AGONISTS HOFFMANN LA ROCHE (CH) 2008-07-09 EP claimed