SCHEMBL5044496

SCHEMBL5044496

CCCCNC(=O)Oc1cc(-c2csc(-c3ccc(C)cc3)n2)n(CC2CCCCC2)c1C

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ATP4A P20648 2/20 0.37
ATP4B P51164 2/20 0.37
LMNA P02545 2/20 0.37
MGLL Q99685 3/20 0.36
ALOX5 P09917 1/20 0.35
TP53 P04637 2/20 0.35
MAPT P10636 1/20 0.35
NTMT1 Q9BV86 1/20 0.34
CDC25A P30304 1/20 0.34
CDC25B P30305 1/20 0.34
CDC25C P30307 1/20 0.34
DUSP3 P51452 1/20 0.34
KLKB1 P03952 1/20 0.34
KLK1 P06870 1/20 0.34
CTSK P43235 1/20 0.34
RORC P51449 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5047889 0.95 MGLL (0.36) LMNAMGLLALOX5TP53MAPT
SCHEMBL5044102 0.94 MAPT (0.40) ATP4AATP4BTP53MAPT
SCHEMBL5040330 0.94 NTMT1 (0.40) LMNAMGLLALOX5TP53NTMT1
SCHEMBL5048696 0.93 CDC25A (0.43) ATP4AATP4BLMNAMGLLTP53
SCHEMBL5039575 0.91 AR (0.43) MGLLALOX5MAPT
SCHEMBL5044042 0.91 CDC25A (0.42) ATP4AATP4BLMNAMGLLTP53
SCHEMBL5047653 0.91 ATP4A (0.38) ATP4AATP4BMGLLTP53MAPT
SCHEMBL5047923 0.89 ATP4A (0.38) ATP4AATP4BLMNAMGLLTP53
SCHEMBL5049183 0.89 NPC1 (0.40) LMNAMAPT
SCHEMBL5133506 0.89 CPT2 (0.40) MGLLCDC25ACDC25BCDC25CDUSP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583762-B1 PYRROLYL-THIAZOLES AND THEIR USE AS CB 1 RECEPTOR INVERSE AGONISTS HOFFMANN LA ROCHE (CH) 2008-07-09 EP claimed