SCHEMBL5047889

SCHEMBL5047889

CCCCNC(=O)Oc1cc(-c2csc(-c3ccc(CC)cc3)n2)n(CC2CCCCC2)c1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 3/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ALOX5 P09917 1/20 0.35
AVPR1B P47901 4/20 0.34
FKBP1A P62942 1/20 0.34
CDC25A P30304 1/20 0.34
CDC25B P30305 1/20 0.34
CDC25C P30307 1/20 0.34
DUSP3 P51452 1/20 0.34
MAPT P10636 2/20 0.34
NPC1 O15118 1/20 0.34
PKM P14618 1/20 0.34
RAB9A P51151 1/20 0.34
CTSK P43235 1/20 0.34
LMNA P02545 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
HTR2A P28223 2/20 0.33
HTR2C P28335 2/20 0.33
SLC6A4 P31645 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5044496 0.95 ATP4A (0.37) MGLLALOX5CDC25ACDC25BCDC25C
SCHEMBL5040330 0.93 NTMT1 (0.40) MGLLALOX5AVPR1BNPC1RAB9A
SCHEMBL5044102 0.93 MAPT (0.40) MAPTNPC1RAB9AHTR2AHTR2C
SCHEMBL5048696 0.92 CDC25A (0.43) MGLLMEN1KMT2AAVPR1BCDC25A
SCHEMBL5039575 0.90 AR (0.43) MGLLMEN1KMT2AALOX5MAPT
SCHEMBL5044042 0.90 CDC25A (0.42) MGLLMEN1KMT2AAVPR1BCDC25A
SCHEMBL5047923 0.89 ATP4A (0.38) MGLLAVPR1BCDC25ACDC25BCDC25C
SCHEMBL5047653 0.89 ATP4A (0.38) MGLLAVPR1BCDC25ACDC25BCDC25C
SCHEMBL5049183 0.88 NPC1 (0.40) MEN1KMT2AMAPTNPC1RAB9A
SCHEMBL5133506 0.88 CPT2 (0.40) MGLLCDC25ACDC25BCDC25CDUSP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583762-B1 PYRROLYL-THIAZOLES AND THEIR USE AS CB 1 RECEPTOR INVERSE AGONISTS HOFFMANN LA ROCHE (CH) 2008-07-09 EP claimed