SCHEMBL5048696

SCHEMBL5048696

CCCCNC(=O)Oc1cc(-c2csc(-c3ccc(OC)cc3)n2)n(CC2CCCCC2)c1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC25A P30304 2/20 0.43
CDC25B P30305 2/20 0.43
CDC25C P30307 2/20 0.43
DUSP3 P51452 2/20 0.43
MAPT P10636 3/20 0.41
TP53 P04637 1/20 0.41
ATP4A P20648 3/20 0.39
ATP4B P51164 3/20 0.39
OXTR P30559 2/20 0.39
AVPR1A P37288 2/20 0.39
AVPR1B P47901 2/20 0.39
MGLL Q99685 2/20 0.39
TDP1 Q9NUW8 1/20 0.38
KLKB1 P03952 1/20 0.37
ALDH1A1 P00352 2/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
KDM4E B2RXH2 1/20 0.37
KMT2A Q03164 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5044042 0.98 CDC25A (0.42) CDC25ACDC25BCDC25CDUSP3MAPT
SCHEMBL5047653 0.93 ATP4A (0.38) CDC25ACDC25BCDC25CDUSP3MAPT
SCHEMBL5044496 0.93 ATP4A (0.37) CDC25ACDC25BCDC25CDUSP3MAPT
SCHEMBL5047889 0.92 MGLL (0.36) CDC25ACDC25BCDC25CDUSP3MAPT
SCHEMBL5040330 0.92 NTMT1 (0.40) TP53AVPR1BMGLLNPC1RAB9A
SCHEMBL5044102 0.92 MAPT (0.40) MAPTTP53ATP4AATP4BALDH1A1
SCHEMBL5039914 0.91 CDC25A (0.45) CDC25ACDC25BCDC25CDUSP3MAPT
SCHEMBL5047923 0.90 ATP4A (0.38) CDC25ACDC25BCDC25CDUSP3MAPT
SCHEMBL5133506 0.90 CPT2 (0.40) CDC25ACDC25BCDC25CDUSP3MGLL
SCHEMBL5048642 0.89 CDC25A (0.44) CDC25ACDC25BCDC25CDUSP3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583762-B1 PYRROLYL-THIAZOLES AND THEIR USE AS CB 1 RECEPTOR INVERSE AGONISTS HOFFMANN LA ROCHE (CH) 2008-07-09 EP claimed