SCHEMBL5049183

SCHEMBL5049183

CCCCNC(=O)Oc1cc(-c2csc(-c3ccc4c(c3)OCO4)n2)n(CC2CCCCC2)c1C

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.40
RAB9A P51151 5/20 0.40
TGFBR1 P36897 8/20 0.39
HPGD P15428 2/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPK1 P28482 1/20 0.37
KCNQ1 P51787 1/20 0.36
LMNA P02545 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAPT P10636 1/20 0.36
CPT2 P23786 1/20 0.35
CPT1A P50416 1/20 0.35
USP2 O75604 1/20 0.35
KDM4E B2RXH2 1/20 0.34
CLK1 P49759 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5043754 0.90 CLK1 (0.45) NPC1RAB9AALDH1A1KMT2ASMN1; SMN2
SCHEMBL5044496 0.89 ATP4A (0.37) LMNAMAPT
SCHEMBL5047889 0.88 MGLL (0.36) NPC1RAB9ALMNAKMT2AMEN1
SCHEMBL4425161 0.88 RAB9A (0.43) NPC1RAB9AHPGDALDH1A1MAPK1
SCHEMBL5039387 0.88 NPC1 (0.47) NPC1RAB9ATGFBR1HPGDALDH1A1
SCHEMBL5044102 0.88 MAPT (0.40) NPC1RAB9AHPGDALDH1A1SMN1; SMN2
SCHEMBL5040330 0.88 NTMT1 (0.40) NPC1RAB9ALMNASMN1; SMN2CPT1A
SCHEMBL5048696 0.87 CDC25A (0.43) NPC1RAB9AHPGDALDH1A1KCNQ1
SCHEMBL5039575 0.85 AR (0.43) RAB9AALDH1A1MAPK1KMT2AMEN1
SCHEMBL5044042 0.85 CDC25A (0.42) NPC1RAB9AALDH1A1KCNQ1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583762-B1 PYRROLYL-THIAZOLES AND THEIR USE AS CB 1 RECEPTOR INVERSE AGONISTS HOFFMANN LA ROCHE (CH) 2008-07-09 EP claimed