Butein

Butein

SCHEMBL505501

O=C(C=Cc1ccc(O)c(O)c1)c1ccc(O)cc1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 1.00
MEN1 O00255 5/20 1.00
NFKB1 P19838 4/20 1.00
NFKB2 Q00653 3/20 1.00
RELA Q04206 3/20 1.00
AKR1B1 P15121 2/20 1.00
HSD17B2 P37059 2/20 1.00
EGFR P00533 1/20 1.00
SRC P12931 1/20 1.00
CDK2 P24941 1/20 1.00
PIK3CA P42336 1/20 1.00
HDAC6 Q9UBN7 1/20 1.00
CYP3A4 P08684 4/20 0.79
TDP1 Q9NUW8 4/20 0.79
MAPT P10636 4/20 0.79
MAPK1 P28482 4/20 0.79
HPGD P15428 3/20 0.79
ALOX15 P16050 3/20 0.79
CYP2C9 P11712 2/20 0.79
CYP2C19 P33261 2/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Butein SCHEMBL29724857 1.00 KMT2A (1.00) KMT2AMEN1NFKB1NFKB2RELA
Butein SCHEMBL243647 1.00 KMT2A (1.00) KMT2AMEN1NFKB1NFKB2RELA
Butein SCHEMBL30383523 1.00 KMT2A (1.00) KMT2AMEN1NFKB1NFKB2RELA
Butein SCHEMBL243646 1.00 KMT2A (1.00) KMT2AMEN1NFKB1NFKB2RELA
Butein SCHEMBL139243 1.00 KMT2A (1.00) KMT2AMEN1NFKB1NFKB2RELA
Butein SCHEMBL25202104 1.00 KMT2A (1.00) KMT2AMEN1NFKB1NFKB2RELA
Butein SCHEMBL25200377 0.98 KMT2A (0.97) KMT2AMEN1NFKB1NFKB2RELA
SCHEMBL25208375 0.90 MEN1 (0.96) KMT2AMEN1NFKB1NFKB2RELA
Butein SCHEMBL25209583 0.89 KMT2A (0.80) KMT2AMEN1NFKB1NFKB2RELA
Butein SCHEMBL1706409 0.89 KMT2A (0.80) KMT2AMEN1NFKB1NFKB2RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 236 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114642695-A Big data traditional Chinese medicine composition for regulating and controlling prostate cancer 华子昂 2022-06-21 CN claimed
US-10588854-B2 Polymer implants for treatment of metabolic disorders UNIVERSITY OF SOUTH CAROLINA (US) 2020-03-17 US claimed
US-20190000749-A1 Polymer Implants for Treatment of Metabolic Disorders NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2019-01-03 US claimed
US-9828407-B2 Water soluble and activable phenolic derivatives with dermocosmetic and therapeutic applications and process for preparing said derivatives LIBRAGEN (FR) 2017-11-28 US claimed
US-20140088030-A1 WATER SOLUBLE AND ACTIVABLE PHENOLICS DERIVATIVES WITH DERMOCOSMETIC AND THERAPEUTIC APPLICATIONS AND PROCESS FOR PREPARING SAID DERIVATIVES LIBRAGEN (FR) 2014-03-27 US claimed
EP-1888174-B1 USE OF CHALCONES FOR THE TREATMENT OF VIRAL DISORDERS JOHNSON & JOHNSON CONSUMER (US) 2012-02-22 EP claimed
US-20100056482-A1 Calixarene Derivatives as Anticancer Agent CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE-CNRS (FR) 2010-03-04 US claimed
EP-1888174-A1 USE OF CHALCONES FOR THE TREATMENT OF VIRAL DISORDERS Johnson and Johnson Consumer Companies, Inc. (US) 2008-02-20 EP claimed
WO-2006127539-A1 USE OF CHALCONES FOR THE TREATMENT OF VIRAL DISORDERS JOHNSON & JOHNSON CONSUMER COMPANIES, INC. (US) 2006-11-30 WO claimed
US-20060270614-A1 Use of chalcones for the treatment of viral disorders JOHNSON & JOHNSON CONSUMER COMPANIES, INC. 2006-11-30 US claimed
WO-2005004814-A2 SIRT1 AND GENETIC DISORDERS ELIXIR PHARMACEUTICALS, INC. (US) 2005-01-20 WO claimed
WO-1995006628-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES OR BACTERIA STATENS SERUMINSTITUT (DK) 1995-03-09 WO claimed
EP-0399051-B1 POLYVALENT ANTIINFLAMMATORY AGENT DAINIPPON INK & CHEMICALS (JP) 1994-05-11 EP claimed
US-5234951-A Anti-ulcer agent comprising chalcone derivative TSUMURA JUNTENDO, INC. (JP) 1993-08-10 US claimed
US-5109025-A Use of 2',3,4,4'-tetrahydroxychalcone (butein) DAINIPPON INK AND CHEMICALS, INC. (JP) 1992-04-28 US claimed
EP-0399051-A1 POLYVALENT ANTIINFLAMMATORY AGENT DAINIPPON INK AND CHEMICALS, INC. (JP) 1990-11-28 EP claimed
EP-0292576-A1 ANTI-ULCEROUS AGENT CONTAINING CHALCONE DERIVATIVE AS EFFECTIVE INGREDIENT AND NOVEL CHALCONE DERIVATIVES TSUMURA & CO. (JP) 1988-11-30 EP claimed
JP-63010720-A None JP disclosed
EP-0292576-A1 ANTI-ULCEROUS AGENT CONTAINING CHALCONE DERIVATIVE AS EFFECTIVE INGREDIENT AND NOVEL CHALCONE DERIVATIVES TSUMURA & CO. (JP) 1988-11-30 EP disclosed
JP-S6310720-A 5-LIPOXYGENASE INHIBITOR AND ANTI-ALLERGIC AGENT NIPPON KAYAKU CO LTD 1988-01-18 JP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10588854-B2 Polymer implants for treatment of metabolic disorders LRBA, FABP4, APMAP KMT2A 1073/4885MEN1 3428/4885NFKB1 1970/4885
US-20060270614-A1 Use of chalcones for the treatment of viral disorders HAVCR2, HMGB3, EIF2AK2 KMT2A 4014/4885MEN1 3326/4885NFKB1 1144/4885
US-20140088030-A1 WATER SOLUBLE AND ACTIVABLE PHENOLICS DERIVATIVES WITH DERMOCOSMETIC AND THERAPEUTIC APPLICATIONS AND PROCESS FOR PREPARING SAID DERIVATIVES UGGT1, TYR, G6PD KMT2A 1919/4885MEN1 4300/4885NFKB1 832/4885
US-20100056482-A1 Calixarene Derivatives as Anticancer Agent CALU, CALR, CALD1 KMT2A 4793/4885MEN1 4432/4885NFKB1 1305/4885
US-20190000749-A1 Polymer Implants for Treatment of Metabolic Disorders LRBA, FABP4, APMAP KMT2A 1073/4885MEN1 3428/4885NFKB1 1970/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.