SCHEMBL5070532

SCHEMBL5070532

Cc1ccc(C(C)C(C(N)=O)P(=O)(O)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.43
REN P00797 3/20 0.43
CTSS P25774 2/20 0.42
CTSL P07711 1/20 0.42
CTSB P07858 1/20 0.42
CTSK P43235 1/20 0.42
ECE1 P42892 1/20 0.42
KLK5 Q9Y337 1/20 0.41
ACE P12821 1/20 0.41
MMP8 P22894 1/20 0.41
MMP14 P50281 1/20 0.41
PSEN1 P49768 4/20 0.40
PSEN2 P49810 4/20 0.40
APH1B Q8WW43 4/20 0.40
NCSTN Q92542 4/20 0.40
APH1A Q96BI3 4/20 0.40
PSENEN Q9NZ42 4/20 0.40
APP P05067 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5070534 0.79 ECE1 (0.48) ATMCTSSCTSLCTSBCTSK
SCHEMBL5070528 0.74 ECE1 (0.48) ATMCTSSCTSLCTSBCTSK
SCHEMBL5135601 0.74 ECE1 (0.48) ATMCTSSCTSLCTSBCTSK
SCHEMBL5069554 0.73 ECE1 (0.48) RENCTSSCTSLCTSBCTSK
SCHEMBL5041973 0.73 ALDH1A1 (0.49) ATMCTSSCTSLCTSBCTSK
SCHEMBL5071371 0.72 ECE1 (0.55) ECE1
SCHEMBL5134614 0.71 ECE1 (0.51) ECE1MMP8MMP14
SCHEMBL4420859 0.71 REN (0.67) ATMRENCTSSCTSLCTSB
SCHEMBL7618822 0.71 REN (0.67) ATMRENCTSSCTSLCTSB
SCHEMBL2173588 0.71 REN (0.67) ATMRENCTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1685142-B1 PHOSPHINIC ACID DERIVATIVES, BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE HOFFMANN LA ROCHE (CH) 2008-01-09 EP disclosed