SCHEMBL5072151

SCHEMBL5072151

[O]c1cc(Br)c(Oc2ccc3nc(O)cc(O)c3c2)c(Br)c1

nearest known ligand 0.40

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
THRB P10828 15/20 0.40
THRA P10827 13/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5072159 0.89 THRB (0.39) THRBTHRA
SCHEMBL3128285 0.83 THRB (0.43) THRBTHRA
SCHEMBL5072132 0.76 NT5E (0.35) THRBTHRA
SCHEMBL5076608 0.73 KDM4E (0.41) THRBTHRA
SCHEMBL5072131 0.72 L3MBTL1 (0.38) THRBTHRA
SCHEMBL6104751 0.71 KDM4E (0.50)
SCHEMBL3140938 0.71 THRA (0.46) THRBTHRA
SCHEMBL5074424 0.69 CYP1A2 (0.44) THRBTHRA
SCHEMBL6089328 0.69 HTT (0.44)
SCHEMBL5072134 0.68 ESR1 (0.38) THRBTHRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899309-A1 HETEROCYCLIC COMPOUNDS AS AGONISTS FOR THE THYROID RECEPTOR KARO BIO AB (SE) 2008-03-19 EP disclosed
WO-2007003419-A1 HETEROCYCLIC COMPOUNDS AS AGONISTS FOR THE THYROID RECEPTOR KARO BIO AB (SE) 2007-01-11 WO disclosed