SCHEMBL5082572

SCHEMBL5082572

COc1c(C=O)c(OC)c(OC)c(OC)c1OC

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 4/20 0.38
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
ERN1 O75460 5/20 0.35
ALDH1A1 P00352 5/20 0.35
CYP2A6 P11509 1/20 0.35
PRKDC P78527 1/20 0.34
LCK P06239 1/20 0.34
GLA P06280 1/20 0.34
MAPT P10636 1/20 0.34
THRB P10828 1/20 0.34
LIMK1 P53667 1/20 0.34
LIMK2 P53671 1/20 0.34
TSHR P16473 2/20 0.33
KDM4E B2RXH2 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MCL1 Q07820 1/20 0.32
IMPDH2 P12268 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28363113 0.91 AKR1B1 (0.37) AKR1B1CA1CA2ERN1ALDH1A1
SCHEMBL22568074 0.90 CA1 (0.38) AKR1B1CA1CA2ERN1ALDH1A1
SCHEMBL16093500 0.85 ERN1 (0.40) AKR1B1CA1CA2ERN1ALDH1A1
SCHEMBL3677774 0.84 AKR1B1 (0.38) AKR1B1CA1CA2ERN1ALDH1A1
SCHEMBL3678520 0.82 ALDH1A1 (0.36) AKR1B1CA1CA2ERN1ALDH1A1
SCHEMBL8684241 0.82 PTPN1 (0.41) AKR1B1CA1CA2ERN1ALDH1A1
SCHEMBL9053478 0.82 AKR1B1 (0.31) AKR1B1
SCHEMBL23917711 0.78 ERN1 (0.42) AKR1B1CA1CA2ERN1ALDH1A1
SCHEMBL7959993 0.78 CA1 (0.32) AKR1B1CA1CA2ERN1ALDH1A1
SCHEMBL4943759 0.77 IMPDH2 (0.42) AKR1B1CA1CA2ERN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080039642-A1 Practical, Cost-Effective Synthesis of Chloromethylated 1, 4-Benzoquinones ZYMES, LLC 2008-02-14 US disclosed
CN-101061085-A A practical, cost-effective method for synthesizing chloromethylated 1, 4-benzoquinones ZYMES LLC (US) 2007-10-24 CN disclosed
WO-2006032425-A2 A PRACTICAL, COST-EFFECTIVE SYNTHESIS OF CHLOROMETHYLATED 1,4-BENZOQUINONES ZYMES, LLC (US) 2006-03-30 WO disclosed
EP-1640355-A1 A practical, cost-effective synthesis of chloromethylated 1,4- benzoquinones BASF AKTIENGESELLSCHAFT (DE) 2006-03-29 EP disclosed
CN-1030415-A Saturated heterocycle carboxamide derivatives and its preparation method YAMANOUCHI PHARMA CO LTD (JP) 1989-01-18 CN disclosed
US-4267344-A 3-PENTA/ALKOXY/BENZYL-; -XANTHYL-, -THIOXANTHYL-, OR -SELENOXANTHYLOXAZOLIDINE-2,5-DIONES PROTEINKEMISK INSTITUT. TILKNYTTET AKADEMIET FOR DE TEKNISKE VIDENSKABER (DK) 1981-05-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080039642-A1 Practical, Cost-Effective Synthesis of Chloromethylated 1, 4-Benzoquinones NDUFA10, NDUFB10, NDUFA5 AKR1B1 659/4885CA1 3987/4885CA2 2696/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.