SCHEMBL5088809

SCHEMBL5088809

O=c1ccc(Cl)nn1C(F)F

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.31
ALDH1A1 P00352 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10072113 0.79 BMPR1B (0.34) KDM4EALDH1A1SMN1; SMN2KMT2A
SCHEMBL17723653 0.75
SCHEMBL10072451 0.73 L3MBTL1 (0.38) KDM4EALDH1A1SMN1; SMN2KMT2A
SCHEMBL29313307 0.71
SCHEMBL29892424 0.71 TP53 (0.34) KDM4EALDH1A1SMN1; SMN2KMT2A
SCHEMBL2464256 0.67
SCHEMBL13660699 0.67
SCHEMBL958356 0.67
Bicarbonate SCHEMBL23649996 0.67 L3MBTL1 (0.39) KDM4EALDH1A1SMN1; SMN2KMT2A
SCHEMBL25261881 0.64 ALDH1A1 (0.36) KDM4EALDH1A1SMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12612372-B2 Oxopyridazinyl-phenyl-carbonohydrazonoyl dicyanide compound and use thereof KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2026-04-28 US disclosed
US-20230278963-A1 NOVEL OXOPYRIDAZINYL-PHENYL-CARBONOHYDRAZONOYL DICYANIDE COMPOUND AND USE THEREOF KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2023-09-07 US disclosed
EP-4169909-A1 NOVEL OXOPYRIDAZINYL-PHENYL-CARBONOHYDRAZONOYL DICYANIDE COMPOUND AND USE THEREOF Korea Institute of Science and Technology (KR) 2023-04-26 EP disclosed
CN-115867279-A Novel oxopyridazinyl-phenyl-carbohydrazone acyldinitrile compounds and use thereof 韩国科学技术研究院 2023-03-28 CN disclosed
US-7419979-B2 Derivatives of 6-{4-[4-(1H-indole-2-sulphonyl)-piperazin-1-carbonyl-phenyl]}pyradizin-3-one ASTRAZENECA AB (SE) 2008-09-02 US disclosed
US-20070135441-A1 New derivatives of 6-{4-[4-(1h-indole-2-sulphonyl)-piperazin-1-carbonyl-phenyl]}pyradizin-3-one ASTRAZENECA AB (SE) 2007-06-14 US disclosed
CN-1905883-A Novel derivatives of 6- { 4- [ 4- (1H-indole-2-sulfonyl) -piperazine-1-carbonyl-phenyl ] } pyridazin-3-one ASTRAZENECA AB (SE) 2007-01-31 CN disclosed
EP-1706120-A1 NEW DERIVATIVES OF 6- 4 4 - 1 H - INDOLE-2-SULPHONYL)-PIPERA ZIN-1-CARBONYL-PHENYL PYRADIZIN-3-ONE AstraZeneca AB (SE) 2006-10-04 EP disclosed
WO-2005065688-A1 NEW DERIVATIVES OF 6-4{4-[1H-INDOLE-2-SULPHONYL)-PIPERAZIN-1-CARBONYL-PHENYL]}PYRADIZIN-3-ONE ASTRAZENECA AB (SE) 2005-07-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12612372-B2 Oxopyridazinyl-phenyl-carbonohydrazonoyl dicyanide compound and use thereof MAPT, MAP2, MAP1B KDM4E 1078/4885ALDH1A1 3523/4885SMN1; SMN2 87/4885
US-20230278963-A1 NOVEL OXOPYRIDAZINYL-PHENYL-CARBONOHYDRAZONOYL DICYANIDE COMPOUND AND USE THEREOF DPP4, QDPR, DPYD KDM4E 2828/4885ALDH1A1 431/4885SMN1; SMN2 4686/4885
US-20070135441-A1 New derivatives of 6-{4-[4-(1h-indole-2-sulphonyl)-piperazin-1-carbonyl-phenyl]}pyradizin-3-one HTR7, TRPC7, HRH4 KDM4E 2216/4885ALDH1A1 1369/4885SMN1; SMN2 4623/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.