SCHEMBL5117818

SCHEMBL5117818

O=C(OCc1ccccc1)[C@@H](O)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.55
MAPK1 P28482 2/20 0.53
TDP1 Q9NUW8 2/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
SLC6A2 P23975 1/20 0.53
SLC6A3 Q01959 1/20 0.53
KMT2A Q03164 1/20 0.53
LMNA P02545 5/20 0.52
LTA4H P09960 1/20 0.50
LAP3 P28838 1/20 0.50
HCAR2 Q8TDS4 1/20 0.49
CES2 O00748 1/20 0.47
CES1 P23141 1/20 0.47
ATM Q13315 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL536227 1.00 ALDH1A1 (0.55) ALDH1A1MAPK1TDP1L3MBTL1SLC6A2
SCHEMBL2231648 1.00 ALDH1A1 (0.55) ALDH1A1MAPK1TDP1L3MBTL1SLC6A2
SCHEMBL10727982 0.91 LMNA (0.57) ALDH1A1MAPK1TDP1L3MBTL1SLC6A2
SCHEMBL10727978 0.91 LMNA (0.57) ALDH1A1MAPK1TDP1L3MBTL1SLC6A2
SCHEMBL11182822 0.88 L3MBTL1 (0.50) ALDH1A1MAPK1TDP1L3MBTL1SLC6A2
SCHEMBL3736834 0.85 ATM (0.65) ALDH1A1TDP1LTA4HLAP3ATM
SCHEMBL22615678 0.85 ATM (0.65) ALDH1A1TDP1LTA4HLAP3ATM
SCHEMBL11845149 0.84 L3MBTL1 (0.46) ALDH1A1MAPK1TDP1L3MBTL1SLC6A2
SCHEMBL8792364 0.84 PTGS1 (0.52) ALDH1A1SLC6A2LMNALTA4HLAP3
Mandelic Acid, Methyl Ester SCHEMBL7704691 0.83 ALDH1A1 (0.50) ALDH1A1MAPK1TDP1L3MBTL1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102791693-B Hepatitis c virus inhibitors BRISTOL-MYERS SQUIBB CO. (US) 2016-04-13 CN disclosed
CN-104072486-B As the connection-1H-benzoglyoxaline of hepatitis C virus inhibitors SQUIBB BRISTOL MYERS CO. (US) 2016-04-06 CN disclosed
CN-101998954-B Conformationally restricted biphenyl derivatives for use as hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2015-06-03 CN disclosed
CN-102459250-B Hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2015-05-06 CN disclosed
CN-102448956-B Hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2015-05-06 CN disclosed
CN-104447707-A Hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2015-03-25 CN disclosed
CN-102459281-B Hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2015-03-11 CN disclosed
CN-101558059-B Hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2014-12-03 CN disclosed
CN-102378762-B Hepatitis c virus inhibitors BRISTOL-MYERS SQUIBB CO. (US) 2014-10-29 CN disclosed
CN-102227407-B Hepatitis c virus inhibitors BRISTOL-MYERS SQUIBB CO. (US) 2014-10-22 CN disclosed
CN-102015692-A Heterocyclic derivatives as hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2011-04-13 CN disclosed
CN-102007122-A Imidazolyl biphenyl imidazoles as hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2011-04-06 CN disclosed
CN-101998954-A Conformationally restricted biphenyl derivatives for use as hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2011-03-30 CN disclosed
CN-101998952-A Hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2011-03-30 CN disclosed
CN-101754966-A Hepatitis c virus inhibitors BRISTOL MYERS SQUIBB CO 2010-06-23 CN disclosed
CN-101558059-A Hepatitis C virus inhibitors BRISTOL MYERS SQUIBB CO (US) 2009-10-14 CN disclosed
US-20080146602-A1 Thienopyridine Derivatives, Production Method and Use Thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-06-19 US disclosed
EP-1751167-A1 THIENOPYRIDINE DERIVATIVES, PRODUCTION METHOD AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-02-14 EP disclosed
WO-2005111046-A1 THIENOPYRIDINE DERIVATIVES, PRODUCTION METHOD AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-11-24 WO disclosed
EP-0554455-A1 OPTICALLY ACTIVE INTERMEDIATE AND PRODUCTION THEREOF SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1993-08-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080146602-A1 Thienopyridine Derivatives, Production Method and Use Thereof IL4, IL5, TSLP ALDH1A1 1425/4885MAPK1 423/4885TDP1 2214/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.