SCHEMBL5135987

SCHEMBL5135987

CCCCn1c(-c2ccccc2)nc(-c2ccccc2)c1CC(NCc1ccc2c(c1)CCN2C(=O)OCC)c1ccc(OC(F)F)cc1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.37
POLB P06746 2/20 0.37
LMNA P02545 6/20 0.35
MAPT P10636 6/20 0.35
ALDH1A1 P00352 1/20 0.34
HTT P42858 1/20 0.34
ROCK1 Q13464 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1913061 0.85 C5AR1 (0.38) TP53POLBLMNAMAPTALDH1A1
SCHEMBL5135107 0.77 C5AR1 (0.47) TP53POLBLMNAMAPTALDH1A1
SCHEMBL5138076 0.77 AGTR1 (0.36)
SCHEMBL5137318 0.76 PIN1 (0.36) ALDH1A1HTT
SCHEMBL5136239 0.74 L3MBTL1 (0.34) LMNAALDH1A1HTT
SCHEMBL648864 0.74 C5AR1 (0.41) ALDH1A1HTT
SCHEMBL5136020 0.74 PTGER4 (0.41) ALDH1A1
SCHEMBL5135264 0.73 ALDH1A1 (0.31) ALDH1A1HTT
SCHEMBL1913060 0.72 C5AR1 (0.56) POLBLMNAMAPTALDH1A1HTT
SCHEMBL5136195 0.72 CA1 (0.33) POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490044-A4 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORP (US) 2008-04-16 EP disclosed
EP-1490044-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2004-12-29 EP disclosed
WO-2003084524-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2003-10-16 WO disclosed