SCHEMBL5138076

SCHEMBL5138076

CCCCn1c(-c2ccccc2)nc(Cl)c1CC(NCc1ccc(C(=O)O)cc1)c1ccc(OC(F)F)cc1

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 2/20 0.36
AGTR2 P50052 2/20 0.36
PLA2G4A P47712 1/20 0.36
PIN1 Q13526 2/20 0.36
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5137318 0.90 PIN1 (0.36) PLA2G4APIN1HDAC1HDAC6
SCHEMBL5136239 0.84 L3MBTL1 (0.34) HDAC1HDAC6
SCHEMBL648619 0.83 AGTR1 (0.40) AGTR1AGTR2PLA2G4APIN1
SCHEMBL5135849 0.83 MDM2 (0.36) PLA2G4APIN1HDAC1HDAC6
SCHEMBL5136020 0.82 PTGER4 (0.41) PLA2G4APIN1HDAC1
SCHEMBL5072300 0.79 PTGER4 (0.36) HDAC1HDAC6
SCHEMBL5137484 0.77 PTGER4 (0.34) PLA2G4APIN1
SCHEMBL5135987 0.77 TP53 (0.37)
SCHEMBL1913031 0.76 TSHR (0.40)
SCHEMBL1912873 0.74 CRHR1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490044-A4 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORP (US) 2008-04-16 EP disclosed
EP-1490044-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2004-12-29 EP disclosed
WO-2003084524-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2003-10-16 WO disclosed