SCHEMBL5137484

SCHEMBL5137484

CCCCn1c(-c2ccccc2)nc(C(F)(F)F)c1CC(NCc1ccc(C(=O)O)cc1)c1cccc(OC(F)(F)C(F)F)c1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 3/20 0.34
PLA2G4A P47712 1/20 0.34
PIN1 Q13526 5/20 0.33
VCP P55072 1/20 0.33
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
HPGD P15428 2/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
CHRM2 P08172 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5135849 0.94 MDM2 (0.36) PTGER4PLA2G4APIN1VCPKDM4E
SCHEMBL5137318 0.88 PIN1 (0.36) PTGER4PLA2G4APIN1KDM4EALDH1A1
SCHEMBL5136239 0.82 L3MBTL1 (0.34) ALDH1A1
SCHEMBL652150 0.82 CRHR1 (0.38)
SCHEMBL5136020 0.80 PTGER4 (0.41) PTGER4PLA2G4APIN1KDM4EALDH1A1
SCHEMBL650362 0.78 TLR7 (0.37) KDM4EALDH1A1
SCHEMBL5138076 0.77 AGTR1 (0.36) PLA2G4APIN1
SCHEMBL651143 0.77 CRHR1 (0.37)
SCHEMBL651001 0.76 CRHR1 (0.38) PIN1
SCHEMBL5137377 0.75 PTGS2 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490044-A4 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORP (US) 2008-04-16 EP disclosed
EP-1490044-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2004-12-29 EP disclosed
WO-2003084524-A1 COMBINATION THERAPY FOR THE TREATMENT OF CONDITIONS WITH PATHOGENIC INFLAMMATORY COMPONENTS NEUROGEN CORPORATION (US) 2003-10-16 WO disclosed