SCHEMBL5145833

SCHEMBL5145833

CC1(C)NC(=O)N(CCNc2ncc(-c3ccccc3)c(-c3ccc(-c4ccccc4)s3)n2)C1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
ADORA1 P30542 5/20 0.40
LMNA P02545 3/20 0.38
HTT P42858 2/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.36
ABL1 P00519 1/20 0.35
PTGS2 P35354 1/20 0.35
GAA P10253 2/20 0.34
USP2 O75604 1/20 0.34
TP53 P04637 1/20 0.34
CYP1A2 P05177 1/20 0.34
GLA P06280 1/20 0.34
CYP2C9 P11712 1/20 0.34
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
HSD17B10 Q99714 1/20 0.34
ADORA2A P29274 1/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5149053 0.92 ALDH1A1 (0.41) ALDH1A1ADORA1LMNAHTTTSHR
SCHEMBL5147378 0.85 ADORA1 (0.40) ALDH1A1ADORA1LMNAHTTTSHR
SCHEMBL2980841 0.84 ADORA1 (0.40) ALDH1A1ADORA1LMNATSHRMAPK1
SCHEMBL5147429 0.84 ADORA1 (0.37) ALDH1A1ADORA1LMNAHTTTSHR
SCHEMBL5147485 0.82 RAF1 (0.39) ALDH1A1ADORA1LMNAHTTTSHR
SCHEMBL5145850 0.82 HSD17B1 (0.38) ALDH1A1ADORA1LMNAHTTTSHR
SCHEMBL5179687 0.81 ADORA1 (0.37) ALDH1A1ADORA1ADORA2A
SCHEMBL5147347 0.80 ADORA1 (0.38) ALDH1A1ADORA1HTTSMN1; SMN2ABL1
SCHEMBL5147476 0.80 HSD17B1 (0.39) ALDH1A1ADORA1LMNAHTTTSHR
SCHEMBL5149006 0.79 ADORA1 (0.39) ALDH1A1ADORA1HTTSMN1; SMN2ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831207-A1 AMINOPYRIMIDINE COMPOUNDS AND METHODS OF USE Amgen Inc. (US) 2007-09-12 EP disclosed
WO-2006066172-A1 AMINOPYRIMIDINE COMPOUNDS AND METHODS OF USE AMGEN, INC. (US) 2006-06-22 WO disclosed