SCHEMBL5134124

SCHEMBL5134124

Cc1c(F)c(C2CCNCC2)c(CC2CCCO2)c(F)c1C(N)=O

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.34
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
PARP1 P09874 1/20 0.32
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
HIF1A Q16665 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5146834 0.83 KMT2A (0.32) KMT2AALDH1A1KDM4EMAPTHPGD
SCHEMBL5134530 0.74 PARP1 (0.33) PARP1
SCHEMBL5134331 0.66 RAB9A (0.39) KMT2AALDH1A1KDM4EHPGDRAB9A
SCHEMBL5134122 0.64 PARP1 (0.41) KMT2AKDM4EHPGDPARP1NPC1
SCHEMBL5134806 0.63 PARP2 (0.39) PARP1
SCHEMBL4763827 0.61 PARP1 (0.54) KMT2AALDH1A1KDM4EMAPTHPGD
SCHEMBL5808501 0.58 HTR2C (0.44) KMT2APARP1
SCHEMBL17594488 0.58 GABRA1 (0.34) KMT2APARP1
SCHEMBL1691748 0.57 ALDH1A1 (0.37) KMT2AALDH1A1KDM4EHPGDRAB9A
SCHEMBL30970522 0.57 PARP1 (0.44) KMT2AALDH1A1KDM4EHPGDPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942893-A2 PIPERIDINE GLYCINE TRANSPORTER INHIBITORS Merck & Co., Inc. (US) 2008-07-16 EP disclosed
WO-2007053400-A2 PIPERIDINE GLYCINE TRANSPORTER INHIBITORS MERCK & CO., INC. (US) 2007-05-10 WO disclosed