SCHEMBL5148557

SCHEMBL5148557

CCN(CC)CC1Cc2cc(C)cc(-c3ccc(OC)cc3)c2O1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.38
PRKAB2 O43741 1/20 0.36
PRKAG1 P54619 1/20 0.36
PRKAA2 P54646 1/20 0.36
PRKAA1 Q13131 1/20 0.36
PRKAG3 Q9UGI9 1/20 0.36
PRKAG2 Q9UGJ0 1/20 0.36
PRKAB1 Q9Y478 1/20 0.36
MAPT P10636 3/20 0.35
ALDH1A1 P00352 3/20 0.35
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33
HTT P42858 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MCHR1 Q99705 1/20 0.33
TSPO P30536 2/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6047897 0.86 GSK3B (0.38) DRD2PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL4222368 0.83 PRKAB2 (0.51) DRD2PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL4226616 0.81 AQP1 (0.45) DRD2PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL4226625 0.81 PRKAB2 (0.42) DRD2PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL4596468 0.78 ALDH1A1 (0.42) DRD2MAPTALDH1A1NPC1RAB9A
SCHEMBL4596465 0.77 ALDH1A1 (0.37) DRD2MAPTALDH1A1NPC1RAB9A
SCHEMBL5148555 0.77 DRD2 (0.37) DRD2MAPTALDH1A1HTTTDP1
SCHEMBL4225733 0.75 ALDH1A1 (0.39) MAPTALDH1A1GAAHTTTDP1
SCHEMBL4790525 0.75 AQP1 (0.56) ALDH1A1NPC1RAB9AF2RL3HRH3
SCHEMBL4789302 0.75 AQP1 (0.45) HRH3METAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1871354-A1 TREATMENT OF PAIN Wyeth (US) 2008-01-02 EP disclosed
WO-2006116171-A1 TREATMENT OF PAIN WYETH (US) 2006-11-02 WO disclosed