Known targets — ChEMBL curated mechanism
AGTR1DHFRGABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTNR3C2PBP2XPTGS1PTGS2VKORC1blablaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAftsImrcAmrcBmrdApbp1apbp1bpbp2apbp2bpbp3polthyA
The experimentally established mechanism targets of Potassium Ion. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.
Predicted protein targets (top 6)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | LMNA | P02545 | 2/20 | 0.38 |
| ▸ | KDM4E | B2RXH2 | 1/20 | 0.32 |
| ▸ | DUSP3 | P51452 | 1/20 | 0.32 |
| ▸ | MEN1 | O00255 | 1/20 | 0.32 |
| ▸ | KMT2A | Q03164 | 1/20 | 0.32 |
| ▸ | CA4 | P22748 | 2/20 | 0.31 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL27825801 | 0.77 | OR51E2 (0.40) | LMNAKDM4EDUSP3MEN1KMT2A | |
| SCHEMBL4214657 | 0.76 | PDE4A (0.39) | LMNAKDM4EDUSP3MEN1KMT2A | |
| Cadaverine Tartrate SCHEMBL3039384 | 0.74 | LMNA (0.50) | LMNACA4 | |
| Cadaverine Tartrate SCHEMBL2031625 | 0.74 | LMNA (0.50) | LMNACA4 | |
| SCHEMBL9188798 | 0.71 | LMNA (0.36) | LMNAKDM4EDUSP3MEN1KMT2A | |
| SCHEMBL4836533 | 0.71 | LMNA (0.36) | LMNAKDM4EDUSP3MEN1KMT2A | |
| SCHEMBL10707703 | 0.69 | CA4 (0.38) | LMNACA4 | |
| Glycerin SCHEMBL28637598 | 0.69 | LMNA (0.56) | LMNACA4 | |
| SCHEMBL3808120 | 0.69 | OR51E2 (0.40) | LMNAKDM4EDUSP3MEN1KMT2A | |
| Potassium Ion SCHEMBL27555296 | 0.69 | LMNA (0.44) | LMNAKDM4EDUSP3MEN1KMT2A |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| US-20180327800-A1 | MONOCLONAL ANTIBODY PRODUCTION BY EBV TRANSFORMATION OF B CELLS | INST RES BIOMEDICINE (CH) | 2018-11-15 | — | — | US | disclosed |
| EP-1597280-B2 | MONOCLONAL ANTIBODY PRODUCTION BY EBV TRANSFORMATION OF B CELLS | INST RESEARCH IN BIOMEDICINE (CH) | 2016-08-24 | — | — | EP | disclosed |
| US-20160160258-A1 | MONOCLONAL ANTIBODY PRODUCTION BY EBV TRANSFORMATION OF B CELLS | INSTITUTE FOR RESEARCH IN BIOMEDICINE (CH) | 2016-06-09 | — | — | US | disclosed |
| US-9290786-B2 | Monoclonal antibody production by EBV transformation of B cells | INSTITUTE FOR RESEARCH IN BIOMEDICINE (CH) | 2016-03-22 | — | — | US | disclosed |
| US-20140004123-A1 | MONOCLONAL ANTIBODY PRODUCTION BY EBV TRANSFORMATION OF B CELLS | INSTITUTE FOR RESEARCH IN BIOMEDICINE (CH) | 2014-01-02 | — | — | US | disclosed |
| EP-1597280-B1 | MONOCLONAL ANTIBODY PRODUCTION BY EBV TRANSFORMATION OF B CELLS | INST RESEARCH IN BIOMEDICINE (CH) | 2012-05-02 | — | — | EP | disclosed |
| US-20120027768-A1 | MONOCLONAL ANTIBODY PRODUCTION BY EBV TRANSFORMATION OF B CELLS | INSTITUTE FOR RESEARCH IN BIOMEDICINE (CH) | 2012-02-02 | — | — | US | disclosed |
| US-8071371-B2 | Monoclonal antibody production by EBV transformation of B cells | HUMABS LLC (US) | 2011-12-06 | — | — | US | disclosed |
| EP-2298804-A2 | Monoclonal antibody production by EBV transformation of B cells | Institute for Research in Biomedicine (CH) | 2011-03-23 | — | — | EP | disclosed |
| US-20100021470-A1 | MONOCLONAL ANTIBODY PRODUCTION BY EBV TRANSFORMATION OF B CELLS | INSTITUTE FOR RESEARCH IN BIOMEDICINE (CH) | 2010-01-28 | — | — | US | disclosed |
| EP-1597280-A2 | MONOCLONAL ANTIBODY PRODUCTION BY EBV TRANSFORMATION OF B CELLS | Institute for Research in Biomedicine (CH) | 2005-11-23 | — | — | EP | disclosed |
| WO-2004076677-A2 | MONOCLONAL ANTIBODY PRODUCTION BY EBV TRANSFORMATION OF B CELLS | INSTITUTE FOR RESEARCH IN BIOMEDICINE (CH) | 2004-09-10 | — | — | WO | disclosed |
| EP-0229767-B1 | IMPROVEMENTS RELATING TO THE DETECTION OF VIRUSES AND ANTIBODIES | ROYAL FREE HOSPITAL SCHOOL OF MEDICINE (GB) | 1990-09-26 | — | — | EP | disclosed |
| US-4937199-A | REMOVING INHIBITORY BETAMICROGLOBULIN FROM CLINICAL SAMPLE-HERPES | THE ROYAL FREE HOSPITAL SCHOOL OF MEDICINE (GB) | 1990-06-26 | — | — | US | disclosed |
| EP-0229767-A1 | IMPROVEMENTS RELATING TO THE DETECTION OF VIRUSES AND ANTIBODIES. | ROYAL FREE HOSP SCHOOL MED (GB) | 1987-07-29 | — | — | EP | disclosed |
| WO-1986005593-A1 | IMPROVEMENTS RELATING TO THE DETECTION OF VIRUSES AND ANTIBODIES | THE ROYAL FREE HOSPITAL SCHOOL OF MEDICINE (GB) | 1986-09-25 | — | — | WO | disclosed |