SCHEMBL5158128

SCHEMBL5158128

CCC(C(=O)O)C(=O)c1ccc(Cl)nc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A12 P48065 1/20 0.37
GABRP O00591 3/20 0.35
GABRD O14764 3/20 0.35
GABRA1 P14867 3/20 0.35
GABRB1 P18505 3/20 0.35
GABRG2 P18507 3/20 0.35
GABRB3 P28472 3/20 0.35
GABRA5 P31644 3/20 0.35
GABRA3 P34903 3/20 0.35
GABRA2 P47869 3/20 0.35
GABRB2 P47870 3/20 0.35
GABRA4 P48169 3/20 0.35
GABRE P78334 3/20 0.35
GABRA6 Q16445 3/20 0.35
GABRG1 Q8N1C3 3/20 0.35
GABRG3 Q99928 3/20 0.35
GABRQ Q9UN88 3/20 0.35
MAPT P10636 2/20 0.33
HTT P42858 2/20 0.33
KLKB1 P03952 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5795930 0.83 SLC6A12 (0.36) SLC6A12GABRPGABRDGABRA1GABRB1
SCHEMBL9144675 0.80 SLC6A12 (0.37) SLC6A12GABRPGABRDGABRA1GABRB1
SCHEMBL29922180 0.79 SLC6A12 (0.36) SLC6A12GABRPGABRDGABRA1GABRB1
SCHEMBL7957108 0.76 SMN1; SMN2 (0.57) L3MBTL1ALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL8801541 0.75 ALDH1A1 (0.38) MAPTHTTKLKB1KLK1L3MBTL1
SCHEMBL5160108 0.75 KEAP1 (0.58) MAPTKDM4EAKR1C3AKR1C2KEAP1
SCHEMBL8548280 0.75 SLC6A12 (0.34) SLC6A12GABRPGABRDGABRA1GABRB1
SCHEMBL8547431 0.74 HSP90AB1 (0.43) SLC6A12GABRPGABRDGABRA1GABRB1
SCHEMBL2082345 0.73 TAS1R3 (0.40) MAPTHTTALDH1A1KDM4ERAB9A
SCHEMBL27446237 0.73 ALDH1A1 (0.37) MAPTHTTL3MBTL1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1340746-B1 Process for the reduction of 3-heteroaryl-3-oxo-propanoic acid derivatives SALTIGO GMBH (DE) 2007-02-28 EP disclosed
EP-1340746-A1 Process for the reduction of 3-heteroaryl-3-oxo-propanoic acid derivatives BAYER AG (DE) 2003-09-03 EP disclosed