SCHEMBL5158380

SCHEMBL5158380

CCCCC(CC)CC(C(=O)O)C(=O)c1cncnc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.37
MAPK1 P28482 3/20 0.37
ALDH1A1 P00352 5/20 0.36
CYP3A4 P08684 3/20 0.36
HCAR2 Q8TDS4 1/20 0.36
HDAC3 O15379 2/20 0.36
HDAC1 Q13547 2/20 0.36
HDAC2 Q92769 2/20 0.36
HDAC4 P56524 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
TSHR P16473 3/20 0.35
LMNA P02545 3/20 0.35
HSD17B10 Q99714 1/20 0.35
AKR1C3 P42330 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5160451 0.84 L3MBTL1 (0.47) ALDH1A1HCAR2HDAC3HDAC1HDAC2
SCHEMBL5160570 0.83 HDAC3 (0.40) CA2MAPK1ALDH1A1CYP3A4HDAC3
SCHEMBL7027705 0.81 ALDH1A1 (0.48) CA2MAPK1ALDH1A1CYP3A4HDAC3
SCHEMBL5162990 0.80 ALDH1A1 (0.36) CA2MAPK1ALDH1A1CYP3A4HDAC3
SCHEMBL7028910 0.79 SLC6A3 (0.45) CA2MAPK1ALDH1A1CYP3A4HDAC3
SCHEMBL5158500 0.78 HCAR2 (0.48) MAPK1ALDH1A1HCAR2AKR1C3AKR1C2
SCHEMBL5163190 0.77 HRH3 (0.44) ALDH1A1HRH4HRH3
SCHEMBL1427672 0.77 CA2 (0.54) CA2MAPK1ALDH1A1CYP3A4TSHR
SCHEMBL5160380 0.76 FAAH (0.43) CA2MAPK1ALDH1A1CYP3A4HDAC3
SCHEMBL5160664 0.76 ALDH1A1 (0.40) CA2MAPK1ALDH1A1CYP3A4HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1340746-B1 Process for the reduction of 3-heteroaryl-3-oxo-propanoic acid derivatives SALTIGO GMBH (DE) 2007-02-28 EP disclosed
EP-1340746-A1 Process for the reduction of 3-heteroaryl-3-oxo-propanoic acid derivatives BAYER AG (DE) 2003-09-03 EP disclosed