SCHEMBL5160129

SCHEMBL5160129

CN(C)C1(CCc2ccccc2)CCC(NC(=O)CCNC(=O)O)CC1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 4/20 0.51
OPRL1 P41146 4/20 0.51
EPHX2 P34913 2/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
EPHX1 P07099 3/20 0.46
NPC1 O15118 1/20 0.44
TP53 P04637 1/20 0.44
TSHR P16473 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KCNA3 P22001 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4867137 0.87 KMT2A (0.48) OPRM1OPRL1EPHX2MEN1KMT2A
SCHEMBL4053293 0.84 KMT2A (0.50) OPRM1OPRL1EPHX2KMT2AEPHX1
SCHEMBL2981366 0.82 EPHX2 (0.50) OPRM1OPRL1EPHX2MEN1KMT2A
SCHEMBL5162372 0.81 RAB9A (0.43) OPRM1OPRL1MEN1KMT2ANPC1
SCHEMBL206731 0.78 HDAC3 (0.51) OPRM1OPRL1EPHX2EPHX1NPC1
SCHEMBL208660 0.78 PLAAT3 (0.46) OPRM1OPRL1EPHX2EPHX1NPC1
SCHEMBL206736 0.77 HPGD (0.48) OPRM1OPRL1EPHX2MEN1KMT2A
SCHEMBL206079 0.76 OPRM1 (0.54) OPRM1OPRL1EPHX2EPHX1
SCHEMBL2985780 0.76 MCHR1 (0.53) EPHX2MEN1KMT2ATP53TSHR
SCHEMBL2972824 0.76 ATF4 (0.59) MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1751090-A1 ACID DERIVATIVES OF SUBSTITUTED CYCLOHEXYL-1,4-DIAMINES Grünenthal GmbH (DE) 2007-02-14 EP disclosed
WO-2005110973-A1 ACID DERIVATIVES OF SUBSTITUTED CYCLOHEXYL-1,4-DIAMINES Grünenthal GmbH (DE) 2005-11-24 WO disclosed