SCHEMBL5166736

SCHEMBL5166736

COc1ccccc1S(=O)(=O)[CH]c1ccccc1OC(C)C

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 12/20 0.51
KCNH2 Q12809 1/20 0.51
PTGES2 Q9H7Z7 2/20 0.49
HTR6 P50406 1/20 0.44
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
ACHE P22303 1/20 0.40
TFEB P19484 1/20 0.40
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5164016 0.73 NFE2L2 (0.48) NFE2L2KCNH2PTGES2HTR6
SCHEMBL29469865 0.71 PTGES2 (0.55) PTGES2ADRA1DADRA1AADRA1BCA1
SCHEMBL2247901 0.71 PTGES2 (0.55) PTGES2ADRA1DADRA1AADRA1BCA1
SCHEMBL5248910 0.71 HTR6 (0.55) NFE2L2KCNH2HTR6CA1CA2
SCHEMBL177279 0.70 ALDH1A1 (0.55) PTGES2ACHEALDH1A1
SCHEMBL13988354 0.69 AR (0.49) NFE2L2PTGES2ACHETFEBALDH1A1
SCHEMBL8711034 0.69 HTR6 (0.53) NFE2L2KCNH2HTR6CA1CA2
SCHEMBL105697 0.69 CA1 (0.65) CA1CA2ACHEALDH1A1
SCHEMBL31433095 0.69 CA1 (0.65) CA1CA2ACHEALDH1A1
SCHEMBL9035206 0.69 ADRA2A (0.54) PTGES2HTR6ADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765332-A2 TRISUBSTITUTED NITROGEN MODULATORS OF TYROSINE PHOSPHATASES Cengent Therapeutics, Inc. (US) 2007-03-28 EP disclosed
WO-2006009876-A2 TRISUBSTITUTED NITROGEN MODULATORS OF TYROSINE PHOSPHATASES CENGENT THERAPEUTICS, INC. (US) 2006-01-26 WO disclosed