SCHEMBL5164016

SCHEMBL5164016

COc1ccccc1S(=O)(=O)[CH]c1ccccc1-c1ccc(C)cc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 10/20 0.48
KCNH2 Q12809 1/20 0.48
HTR6 P50406 1/20 0.44
ACLY P53396 1/20 0.38
PTGES2 Q9H7Z7 1/20 0.38
PTGS1 P23219 2/20 0.38
PTGS2 P35354 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
PTPRC P08575 1/20 0.38
PTPN1 P18031 1/20 0.38
NR1H3 Q13133 1/20 0.37
SYK P43405 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5166736 0.73 NFE2L2 (0.51) NFE2L2KCNH2HTR6PTGES2
SCHEMBL5164020 0.73 TSHR (0.41) HTR6CYP3A4CYP2C9CYP2C19SYK
SCHEMBL4425113 0.72 SYK (0.56) PTPRCPTPN1SYK
SCHEMBL28541778 0.71 HTR6 (0.77) HTR6
SCHEMBL5165214 0.70 MEN1 (0.48)
SCHEMBL21471580 0.70 PTPRC (0.47) PTPRCPTPN1SYK
SCHEMBL7932563 0.69 ERN1 (0.44) NFE2L2SYK
SCHEMBL5248910 0.68 HTR6 (0.55) NFE2L2KCNH2HTR6
SCHEMBL8552729 0.68 CA2 (0.53) PTGES2PTGS1PTGS2CYP2C9
SCHEMBL9693255 0.67 NAMPT (0.45) PTGS2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765332-A2 TRISUBSTITUTED NITROGEN MODULATORS OF TYROSINE PHOSPHATASES Cengent Therapeutics, Inc. (US) 2007-03-28 EP disclosed
WO-2006009876-A2 TRISUBSTITUTED NITROGEN MODULATORS OF TYROSINE PHOSPHATASES CENGENT THERAPEUTICS, INC. (US) 2006-01-26 WO disclosed