SCHEMBL5190765

SCHEMBL5190765

CC(=O)N1CCNC(CC(=O)NCCc2ccc(Cl)cc2)C1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.47
HTR2A P28223 1/20 0.47
MCHR1 Q99705 1/20 0.47
ALDH1A1 P00352 2/20 0.46
MAPT P10636 2/20 0.46
KDM4E B2RXH2 1/20 0.46
LMNA P02545 2/20 0.45
TSHR P16473 1/20 0.43
HSD17B10 Q99714 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
GAA P10253 1/20 0.41
HTT P42858 1/20 0.41
POLB P06746 1/20 0.41
EPHX1 P07099 1/20 0.41
EPHX2 P34913 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5193308 0.86 POLB (0.47) ALDH1A1MAPTKDM4ELMNATSHR
SCHEMBL5193468 0.82 ALDH1A1 (0.52) ALDH1A1MAPTKDM4ELMNAHSD17B10
SCHEMBL5193913 0.79 NPC1 (0.44) ALDH1A1MAPTLMNANPC1RAB9A
SCHEMBL5194854 0.77 NPC1 (0.44) ALDH1A1LMNANPC1RAB9AGAA
SCHEMBL5191071 0.77 LMNA (0.47) MAPTLMNAGAA
SCHEMBL5214027 0.76 NPC1 (0.53) ALDH1A1LMNANPC1RAB9APOLB
SCHEMBL5194022 0.76 ALDH1A1 (0.46) ALDH1A1MAPTKDM4EHSD17B10POLB
SCHEMBL5190984 0.74 ALDH1A1 (0.41) ALDH1A1MAPTKDM4ELMNACYP2C19
SCHEMBL5191129 0.72 CA1 (0.46) ALDH1A1MAPTCYP2C19NPC1RAB9A
SCHEMBL8472774 0.71 EPHX1 (0.54) CHRM1HTR2AMCHR1MAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP disclosed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP disclosed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO disclosed