SCHEMBL5190984

SCHEMBL5190984

CCCNC(=O)N1CCNC(CC(=O)NCCc2ccc(F)c(F)c2)C1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.41
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
KDM4E B2RXH2 3/20 0.39
LMNA P02545 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
CYP2C19 P33261 2/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.37
PARP1 P09874 2/20 0.37
PARP2 Q9UGN5 2/20 0.37
MAPT P10636 1/20 0.37
PTGDR2 Q9Y5Y4 2/20 0.36
CCR3 P51677 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5193913 0.81 NPC1 (0.44) ALDH1A1MEN1KMT2ALMNAHPGD
SCHEMBL5278574 0.75 LMNA (0.48) LMNACCR3
SCHEMBL5190765 0.74 CHRM1 (0.47) ALDH1A1KDM4ELMNACYP2C19MAPT
SCHEMBL5191885 0.74 LMNA (0.44) ALDH1A1MEN1KMT2AKDM4ELMNA
SCHEMBL5193468 0.73 ALDH1A1 (0.52) ALDH1A1MEN1KMT2AKDM4ELMNA
SCHEMBL5194080 0.71 ALDH1A1 (0.46) ALDH1A1MEN1KMT2AKDM4ELMNA
SCHEMBL5213606 0.71 KMT2A (0.60) ALDH1A1MEN1KMT2AKDM4ELMNA
SCHEMBL5192795 0.70 NOS2 (0.49)
SCHEMBL5193560 0.69 CCR2 (0.48) ALDH1A1MEN1KMT2ALMNAMAPT
SCHEMBL5190775 0.69 MAPT (0.49) ALDH1A1MEN1KMT2ALMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP claimed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP claimed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO claimed