SCHEMBL5214027

SCHEMBL5214027

CN1CCNC(CC(=O)NCc2ccc(Cl)cc2)C1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.53
RAB9A P51151 2/20 0.53
ALDH1A1 P00352 3/20 0.48
LMNA P02545 1/20 0.48
POLB P06746 2/20 0.48
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
HPGD P15428 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5194854 0.82 NPC1 (0.44) NPC1RAB9AALDH1A1LMNAPOLB
SCHEMBL5193913 0.82 NPC1 (0.44) NPC1RAB9AALDH1A1LMNAPOLB
SCHEMBL5195403 0.81 HPGD (0.42) NPC1RAB9ALMNAMEN1KMT2A
SCHEMBL5191220 0.79 FAAH (0.51) NPC1RAB9ALMNAPOLBMEN1
SCHEMBL5191129 0.77 CA1 (0.46) NPC1RAB9AALDH1A1POLBMEN1
SCHEMBL5190765 0.76 CHRM1 (0.47) NPC1RAB9AALDH1A1LMNAPOLB
SCHEMBL5192010 0.74 HPGD (0.46) ALDH1A1MEN1KMT2AHPGD
SCHEMBL5193934 0.73 ALDH1A1 (0.53) ALDH1A1LMNAMEN1KMT2AHPGD
SCHEMBL2917177 0.73 REN (0.35) LMNA
SCHEMBL4672942 0.73 RAB9A (0.74) NPC1RAB9AALDH1A1LMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP disclosed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP disclosed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO disclosed