SCHEMBL5194091

SCHEMBL5194091

COc1ccc(CNC(=O)CC2CN(C(=O)Nc3ccccc3)CCN2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 2/20 0.53
RAB9A P51151 2/20 0.51
NPC1 O15118 2/20 0.51
GLA P06280 1/20 0.50
CCR3 P51677 1/20 0.50
MEN1 O00255 4/20 0.48
KMT2A Q03164 4/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
THRB P10828 1/20 0.48
CDK1 P06493 1/20 0.47
IGF1R P08069 1/20 0.47
FGFR1 P11362 1/20 0.47
BRAF P15056 1/20 0.47
FGFR2 P21802 1/20 0.47
FGFR4 P22455 1/20 0.47
FGFR3 P22607 1/20 0.47
JAK1 P23458 1/20 0.47
CDK2 P24941 1/20 0.47
AXL P30530 1/20 0.47
CDK5 Q00535 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5193432 0.95 MAPT (0.50) FAAHRAB9AGLACCR3MEN1
SCHEMBL5193739 0.92 PKM (0.56) RAB9AGLACCR3MEN1KMT2A
SCHEMBL5191220 0.87 FAAH (0.51) FAAHRAB9ANPC1MEN1KMT2A
SCHEMBL5210355 0.87 CCR2 (0.50) RAB9ANPC1CCR3MEN1KMT2A
SCHEMBL5192491 0.82 ALDH1A1 (0.45) NPC1MEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL5208438 0.81 FAAH (0.54) FAAHRAB9ANPC1CCR3MEN1
SCHEMBL5190018 0.81 PKM (0.49) NPC1MEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL5193199 0.80 MAPT (0.55) RAB9ANPC1CCR3MEN1KMT2A
SCHEMBL5193499 0.80 FAAH (0.52) FAAHCCR3MEN1KMT2ASMN1; SMN2
SCHEMBL5190651 0.79 KMT2A (0.42) NPC1MEN1KMT2ASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP claimed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP claimed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO claimed