SCHEMBL5192806

SCHEMBL5192806

CN(C)S(=O)(=O)N1CCNCC1CC(N)=O

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.33
CA1 P00915 4/20 0.33
CA2 P00918 4/20 0.33
CA4 P22748 4/20 0.33
CA9 Q16790 4/20 0.33
ALDH1A1 P00352 1/20 0.33
MMP1 P03956 1/20 0.30
MMP3 P08254 1/20 0.30
MMP7 P09237 1/20 0.30
MMP9 P14780 1/20 0.30
MMP13 P45452 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5191931 0.84 CA1 (0.34) CA1CA2CA4CA9MMP1
SCHEMBL5195643 0.75 MMP8 (0.35) CA1CA2CA4CA9ALDH1A1
SCHEMBL2919209 0.73 TSHR (0.36) CA1CA2CA4CA9
SCHEMBL25154636 0.70 SLC6A1 (0.40) CA1CA2CA4CA9MMP1
SCHEMBL3624075 0.69 CA1 (0.34) CA1CA2CA4CA9
SCHEMBL2917654 0.68 KDM4E (0.37)
SCHEMBL5190158 0.68 PARP1 (0.36) CA1CA2CA4CA9
SCHEMBL5195457 0.66 FHIT (0.34) CA1CA2CA4CA9
SCHEMBL5195326 0.64 LMNA (0.39) CA1CA2CA4CA9
SCHEMBL1087766 0.64 ALOX5AP (0.36) CA1CA2CA4CA9MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP disclosed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP disclosed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO disclosed