SCHEMBL5197846

SCHEMBL5197846

Cn1cc(-c2cc(-c3cn(COCC[Si](C)(C)C)nc3-c3ccccn3)ccc2F)cn1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 4/20 0.39
PIM3 Q86V86 1/20 0.39
PIM2 Q9P1W9 1/20 0.39
FEN1 P39748 5/20 0.38
ALOX5AP P20292 4/20 0.38
TGFBR1 P36897 3/20 0.38
ACVR1B P36896 1/20 0.38
KDR P35968 1/20 0.36
EPHB4 P54760 1/20 0.36
TEK Q02763 1/20 0.36
MET P08581 1/20 0.34
GRM5 P41594 1/20 0.34
MAPK1 P28482 2/20 0.34
CHRM1 P11229 1/20 0.33
ABL1 P00519 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5198347 0.84 DGAT1 (0.35) FEN1ALOX5APTGFBR1GRM5
SCHEMBL5197725 0.83 GABRA2 (0.39) FEN1ALOX5AP
SCHEMBL5198955 0.76 TGFBR1 (0.47) TGFBR1MAPK1
SCHEMBL5199830 0.76 PIM1 (0.50) PIM1PIM3PIM2FEN1ALOX5AP
SCHEMBL5197736 0.74 TGFBR1 (0.42) TGFBR1
SCHEMBL5198600 0.74 DGAT1 (0.41) TGFBR1
SCHEMBL16022794 0.73 GSK3B (0.38) FEN1ALOX5APMET
SCHEMBL30725992 0.73 KDM4E (0.38) TGFBR1GRM5
SCHEMBL5199272 0.72 CNR2 (0.42) TGFBR1
SCHEMBL31074732 0.72 CYP1A2 (0.35) TGFBR1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070275968-A1 Substituted Biphenyl Derivative SANKYO COMPANY, LIMITED (JP) 2007-11-29 US disclosed
EP-1798229-A1 SUBSTITUTED BIPHENYL DERIVATIVE Sankyo Company, Limited (JP) 2007-06-20 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070275968-A1 Substituted Biphenyl Derivative COL2A1, COL1A1, FGFR3 PIM1 4793/4885PIM3 4397/4885PIM2 4679/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.