SCHEMBL5199830

SCHEMBL5199830

Cn1cc(-c2cc(-c3c[nH]nc3-c3ccccn3)ccc2F)cn1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 6/20 0.50
PIM3 Q86V86 1/20 0.50
PIM2 Q9P1W9 1/20 0.50
TGFBR1 P36897 3/20 0.47
ACVR1B P36896 1/20 0.47
ALOX5AP P20292 1/20 0.44
FEN1 P39748 1/20 0.44
MAP4K1 Q92918 2/20 0.41
AXL P30530 2/20 0.39
LRRK2 Q5S007 2/20 0.39
CLK2 P49760 1/20 0.38
CLK3 P49761 1/20 0.38
DYRK1A Q13627 1/20 0.38
KDR P35968 1/20 0.37
EPHB4 P54760 1/20 0.37
TEK Q02763 1/20 0.37
ALK Q9UM73 1/20 0.37
PDK2 Q15119 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24312429 0.86 FEN1 (0.49) PIM1PIM3PIM2TGFBR1ALOX5AP
SCHEMBL5198228 0.84 TGFBR1 (0.52) PIM1TGFBR1ALOX5APFEN1MAP4K1
SCHEMBL5197608 0.76 KDM4E (0.37) PIM1TGFBR1LRRK2
SCHEMBL5197846 0.76 PIM1 (0.39) PIM1PIM3PIM2TGFBR1ACVR1B
SCHEMBL5199408 0.76 PTGS2 (0.46)
SCHEMBL373516 0.74 TGFBR1 (0.59) PIM1TGFBR1MAP4K1AXLCLK2
SCHEMBL5490810 0.73 TGFBR1 (0.54) TGFBR1LRRK2
SCHEMBL23218015 0.73 TGFBR1 (0.59) TGFBR1ALOX5APFEN1KDREPHB4
SCHEMBL5199498 0.72 TGFBR1 (0.56) PIM1PIM3PIM2TGFBR1LRRK2
SCHEMBL29361356 0.72 TGFBR1 (0.70) PIM1TGFBR1FEN1PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070275968-A1 Substituted Biphenyl Derivative SANKYO COMPANY, LIMITED (JP) 2007-11-29 US disclosed
EP-1798229-A1 SUBSTITUTED BIPHENYL DERIVATIVE Sankyo Company, Limited (JP) 2007-06-20 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070275968-A1 Substituted Biphenyl Derivative COL2A1, COL1A1, FGFR3 PIM1 4793/4885PIM3 4397/4885PIM2 4679/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.