SCHEMBL5199846

SCHEMBL5199846

CCCCOC(=O)NC(Cc1ccc(OC)c(OC)c1OC)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.41
KDM4E B2RXH2 4/20 0.40
L3MBTL1 Q9Y468 3/20 0.40
LMNA P02545 2/20 0.40
TSHR P16473 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
ITGB3 P05106 4/20 0.38
ITGA2B P08514 4/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ALOX15 P16050 1/20 0.38
GAA P10253 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
CASP1 P29466 1/20 0.38
HSD17B10 Q99714 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5088784 0.84 ALDH1A1 (0.52) ALDH1A1KDM4ELMNATSHRNPSR1
SCHEMBL5198519 0.81 ALDH1A1 (0.45) ALDH1A1L3MBTL1LMNATSHRNPSR1
SCHEMBL5499791 0.81 LDHA (0.54) ALDH1A1ITGB3ITGA2BMEN1KMT2A
SCHEMBL2675317 0.80 ITGA4 (0.49) KDM4EITGB3ITGA2B
SCHEMBL2675313 0.80 ITGA4 (0.49) KDM4EITGB3ITGA2B
SCHEMBL2149054 0.80 POLB (0.45) ALDH1A1TSHRITGB3ITGA2BALOX15
SCHEMBL2320402 0.77 FPR2 (0.54) ITGB3ITGA2BKMT2A
SCHEMBL8485515 0.77 FPR2 (0.54) ITGB3ITGA2BKMT2A
SCHEMBL7862434 0.76 ALDH1A1 (0.50) ALDH1A1TSHRALOX15GAATDP1
SCHEMBL7378641 0.76 ALDH1A1 (0.54) ALDH1A1LMNATSHRNPSR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1576179-A4 METHODS AND COMPOSITIONS FOR INDUCING APOPTOSIS IN CANCER CELLS IRM LLC (BM) 2007-06-06 EP disclosed
EP-1576179-A2 METHODS AND COMPOSITIONS FOR INDUCING APOPTOSIS IN CANCER CELLS IRM LLC (BM) 2005-09-21 EP disclosed
WO-2004050895-A2 METHODS AND COMPOSITIONS FOR INDUCING APOPTOSIS IN CANCER CELLS IRM LLC (BM) 2004-06-17 WO disclosed
EP-1399468-A1 2-((N-(2-AMINO-3-(HETEROARYL OR ARYL)PROPIONYL)-AMINOACYL)-AMINO)-ALKYLBORONIC ACID DERIVATIVES Novartis AG (CH) 2004-03-24 EP disclosed
WO-2002096933-A1 2-{[N-(2-AMINO-3-(HETEROARYL OR ARYL)PROPIONYL)-AMINOACYL]-AMINO}-ALKYLBORONIC ACID DERIVATIVES NOVARTIS AG (CH) 2002-12-05 WO disclosed