SCHEMBL5200536

SCHEMBL5200536

CCCCc1ccc(OC)c(CC[C@H](O)c2ccccc2)c1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.50
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
SIGMAR1 Q99720 2/20 0.43
HTR1A P08908 1/20 0.43
PPARG P37231 2/20 0.42
PPARA Q07869 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL579636 0.88 ADRB2 (0.50) ADRB2KDM4EALDH1A1HTR1APPARG
SCHEMBL580491 0.88 ADRB2 (0.50) ADRB2KDM4EALDH1A1HTR1APPARG
SCHEMBL6367936 0.79 ALOX5 (0.50) PPARGPPARA
SCHEMBL8534575 0.79 ADRB2 (0.54) ADRB2KDM4EALDH1A1
SCHEMBL5200533 0.79 SIGMAR1 (0.46) SIGMAR1HTR1A
SCHEMBL10235750 0.78 PPARG (0.46) KDM4EALDH1A1PPARGPPARA
SCHEMBL10235726 0.78 PPARG (0.46) KDM4EALDH1A1PPARGPPARA
SCHEMBL580495 0.77 RIPK1 (0.44) ADRB2KDM4EALDH1A1HTR1A
SCHEMBL5198250 0.75 PPARG (0.42) ADRB2SIGMAR1HTR1APPARGPPARA
SCHEMBL5200538 0.75 PPARG (0.42) ADRB2SIGMAR1HTR1APPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633695-A4 SMOOTH MUSCLE SPASMOLYTIC AGENTS BRIDGE PHARMA INC (US) 2007-12-12 EP disclosed
EP-1633695-A2 SMOOTH MUSCLE SPASMOLYTIC AGENTS Bridge Pharma, Inc. (US) 2006-03-15 EP disclosed
WO-2004105692-A2 SMOOTH MUSCLE SPASMOLYTIC AGENTS BRIDGE PHARMA, INC. (US) 2004-12-09 WO disclosed