SCHEMBL5201178

SCHEMBL5201178

CCOC(=O)Cc1ccc(CC(=O)OCC)c(NC2CCN(CCc3ccccc3Cl)CC2)c1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
MAPT P10636 2/20 0.43
SIGMAR1 Q99720 1/20 0.42
HTR4 Q13639 1/20 0.40
KDM4E B2RXH2 2/20 0.40
TSHR P16473 1/20 0.40
KCNH2 Q12809 1/20 0.40
GAA P10253 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HTR1A P08908 1/20 0.39
SLC6A4 P31645 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5201180 0.96 KDM1A (0.42) ALDH1A1MAPTSIGMAR1HTR4TSHR
SCHEMBL5201971 0.89 CACNA1G (0.44) ALDH1A1SIGMAR1KDM4EKCNH2GAA
SCHEMBL5201976 0.85 OPRM1 (0.43) ALDH1A1SIGMAR1KDM4EGAAHSD17B10
SCHEMBL5203921 0.81 CNR1 (0.43) ALDH1A1SIGMAR1KDM4ETSHRKCNH2
SCHEMBL5201928 0.78 SIGMAR1 (0.47) ALDH1A1SIGMAR1GAAHSD17B10HTR1A
SCHEMBL5202261 0.78 CACNA1G (0.44) ALDH1A1KCNH2GAAHSD17B10
SCHEMBL5203925 0.77 CNR1 (0.43) ALDH1A1SIGMAR1KDM4ETSHRGAA
SCHEMBL5202266 0.74 CACNA1G (0.42) ALDH1A1SIGMAR1GAAHSD17B10
SCHEMBL5709511 0.71 SIGMAR1 (0.60) SIGMAR1KCNH2
SCHEMBL5204633 0.71 SIGMAR1 (0.46) ALDH1A1SIGMAR1GAAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1179532-B1 PROCESS FOR THE PRODUCTION OF INDOLE DERIVATIVES AND INTERMEDIATES THEREFOR EISAI R&D MAN CO LTD (JP) 2007-06-13 EP disclosed
US-6573384-B1 1,4-substituted cyclic amine compound which is useful as a pharmaceutical, and an intermediate for the process EISAI CO., LTD. (JP) 2003-06-03 US disclosed
EP-1179532-A1 PROCESS FOR THE PRODUCTION OF INDOLE DERIVATIVES AND INTERMEDIATES THEREFOR Eisai Co., Ltd. (JP) 2002-02-13 EP disclosed