SCHEMBL5201928

SCHEMBL5201928

COC(=O)Cc1ccc(CC(=O)OC)c(NC2CCN(CCc3cccc(Cl)c3)CC2)c1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.47
HTR1A P08908 1/20 0.45
SLC6A4 P31645 1/20 0.45
ALDH1A1 P00352 1/20 0.45
GAA P10253 1/20 0.45
HSD17B10 Q99714 1/20 0.45
CARM1 Q86X55 1/20 0.42
PRMT6 Q96LA8 1/20 0.42
MAPK1 P28482 1/20 0.42
CNR1 P21554 1/20 0.42
OPRM1 P35372 1/20 0.41
CCR5 P51681 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5201931 0.95 SIGMAR1 (0.47) SIGMAR1HTR1ASLC6A4ALDH1A1GAA
SCHEMBL5204629 0.89 SIGMAR1 (0.48) SIGMAR1ALDH1A1GAAHSD17B10CARM1
SCHEMBL5204633 0.85 SIGMAR1 (0.46) SIGMAR1ALDH1A1GAAHSD17B10OPRM1
SCHEMBL5203921 0.81 CNR1 (0.43) SIGMAR1HTR1ASLC6A4ALDH1A1GAA
SCHEMBL5201178 0.78 ALDH1A1 (0.44) SIGMAR1HTR1ASLC6A4ALDH1A1GAA
SCHEMBL5202261 0.75 CACNA1G (0.44) ALDH1A1GAAHSD17B10OPRM1
SCHEMBL5201971 0.75 CACNA1G (0.44) SIGMAR1ALDH1A1GAAHSD17B10MAPK1
SCHEMBL5201180 0.74 KDM1A (0.42) SIGMAR1ALDH1A1GAAHSD17B10OPRM1
SCHEMBL8609753 0.74 SIGMAR1 (0.61) SIGMAR1HTR1AALDH1A1GAAHSD17B10
SCHEMBL13202954 0.73 CARM1 (0.62) SIGMAR1HTR1ASLC6A4ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1179532-B1 PROCESS FOR THE PRODUCTION OF INDOLE DERIVATIVES AND INTERMEDIATES THEREFOR EISAI R&D MAN CO LTD (JP) 2007-06-13 EP disclosed
US-6573384-B1 1,4-substituted cyclic amine compound which is useful as a pharmaceutical, and an intermediate for the process EISAI CO., LTD. (JP) 2003-06-03 US disclosed
EP-1179532-A1 PROCESS FOR THE PRODUCTION OF INDOLE DERIVATIVES AND INTERMEDIATES THEREFOR Eisai Co., Ltd. (JP) 2002-02-13 EP disclosed