SCHEMBL5201976

SCHEMBL5201976

CCOC(=O)Cc1ccc(CC(=O)O)cc1NC1CCN(CCc2ccccc2F)CC1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.43
CACNA1G O43497 1/20 0.42
KDM1A O60341 3/20 0.42
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
POLB P06746 1/20 0.42
GAA P10253 1/20 0.42
HSD17B10 Q99714 1/20 0.42
SIGMAR1 Q99720 4/20 0.41
PTGDR2 Q9Y5Y4 5/20 0.40
CCR3 P51677 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5201971 0.96 CACNA1G (0.44) OPRM1CACNA1GKDM1AALDH1A1KDM4E
SCHEMBL5201180 0.90 KDM1A (0.42) OPRM1KDM1AALDH1A1GAAHSD17B10
SCHEMBL5201178 0.85 ALDH1A1 (0.44) ALDH1A1KDM4EGAAHSD17B10SIGMAR1
SCHEMBL5202266 0.82 CACNA1G (0.42) OPRM1CACNA1GKDM1AALDH1A1GAA
SCHEMBL5204633 0.79 SIGMAR1 (0.46) OPRM1CACNA1GKDM1AALDH1A1GAA
SCHEMBL5201290 0.79 ACACB (0.44) KDM1AALDH1A1POLBHSD17B10PTGDR2
SCHEMBL5203925 0.79 CNR1 (0.43) KDM1AALDH1A1KDM4EGAAHSD17B10
SCHEMBL5202261 0.77 CACNA1G (0.44) OPRM1CACNA1GALDH1A1GAAHSD17B10
SCHEMBL5201931 0.76 SIGMAR1 (0.47) OPRM1ALDH1A1GAAHSD17B10SIGMAR1
SCHEMBL5204629 0.74 SIGMAR1 (0.48) OPRM1CACNA1GALDH1A1GAAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1179532-B1 PROCESS FOR THE PRODUCTION OF INDOLE DERIVATIVES AND INTERMEDIATES THEREFOR EISAI R&D MAN CO LTD (JP) 2007-06-13 EP disclosed
US-6573384-B1 1,4-substituted cyclic amine compound which is useful as a pharmaceutical, and an intermediate for the process EISAI CO., LTD. (JP) 2003-06-03 US disclosed
EP-1179532-A1 PROCESS FOR THE PRODUCTION OF INDOLE DERIVATIVES AND INTERMEDIATES THEREFOR Eisai Co., Ltd. (JP) 2002-02-13 EP disclosed