SCHEMBL5204446

SCHEMBL5204446

Cc1cc(C2CCCN2C(=O)O)nc(-c2ncc[nH]2)n1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 8/20 0.37
UCHL1 P09936 1/20 0.36
USP30 Q70CQ3 1/20 0.36
HCRTR2 O43614 7/20 0.35
GRM5 P41594 4/20 0.35
NOS1 P29475 2/20 0.34
NOS2 P35228 2/20 0.34
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
GCK P35557 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MAPK14 Q16539 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4640604 0.83 AADAT (0.45) KDM4EGCKMEN1KMT2A
SCHEMBL5200371 0.77 NOS1 (0.36) HCRTR1NOS1NOS2
SCHEMBL2637675 0.74 SMN1; SMN2 (0.39) HCRTR1UCHL1USP30HCRTR2KDM4E
SCHEMBL5199947 0.72 HRH3 (0.35) HCRTR1HCRTR2KDM4EALDH1A1MEN1
SCHEMBL934063 0.72 HTR2B (0.42) HCRTR1HCRTR2
SCHEMBL1293292 0.72 HTR2B (0.42) HCRTR1HCRTR2
SCHEMBL5203615 0.71 UCHL1 (0.38) HCRTR1UCHL1USP30HCRTR2GRM5
SCHEMBL4641452 0.71 SCN10A (0.35) HCRTR1HCRTR2
SCHEMBL3566595 0.70 NOS2 (0.59) NOS1NOS2KDM4EALDH1A1MEN1
SCHEMBL5202000 0.70 MEN1 (0.33) HCRTR1HCRTR2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817030-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS Kalypsys, Inc. (US) 2007-08-15 EP disclosed
WO-2007062417-A1 METHODS OF PREPARING 2-IMIDAZOL-1-YL-4-METHYL-6-PYRROLIDIN-2-YL-PYRIMIDINE AND 4-(1-ALKYLPYRROLIDIN-2-YL)-2-(1H-IMIDAZOL-1-YL)-6-METHYLPYRIMIDINE DERIVATIVES KALYPSYS, INC. (US) 2007-05-31 WO disclosed
WO-2006060424-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS KALYPSYS, INC. (US) 2006-06-08 WO disclosed