SCHEMBL5202000

SCHEMBL5202000

Cc1cc(C2CCCCN2)nc(-c2ncc[nH]2)n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2C19 P33261 2/20 0.33
KMT2A Q03164 2/20 0.33
POLB P06746 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNA7 P36544 1/20 0.33
CHRNA4 P43681 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2A6 P11509 1/20 0.33
CYP2C9 P11712 1/20 0.33
AURKA O14965 1/20 0.33
CDC7 O00311 5/20 0.32
CCNE1 P24864 5/20 0.32
CDK2 P24941 5/20 0.32
ROCK1 Q13464 5/20 0.32
DBF4 Q9UBU7 5/20 0.32
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4641452 0.96 SCN10A (0.35) CHRNB2CHRNA7CHRNA4HCRTR1HCRTR2
SCHEMBL5200864 0.73 ADORA2A (0.33)
SCHEMBL5199693 0.71 MAPT (0.34) MEN1KMT2AHCRTR1HCRTR2
SCHEMBL5204446 0.70 HCRTR1 (0.37) MEN1KMT2AHCRTR1HCRTR2
SCHEMBL5200371 0.69 NOS1 (0.36) HCRTR1
SCHEMBL5199466 0.68 LMNA (0.46) MEN1KMT2ASMN1; SMN2ADRA2ANISCH
SCHEMBL6173530 0.67 CHRNB2 (0.45) MEN1CYP2D6CYP2C19KMT2APOLB
SCHEMBL3562054 0.67 NOS2 (0.41) MEN1CYP2D6CYP2C19KMT2APOLB
SCHEMBL3346462 0.65 MEN1 (0.37) MEN1CYP2D6CYP2C19KMT2APOLB
SCHEMBL9026316 0.63 NISCH (0.50) MEN1CYP2D6CYP2C19KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817030-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS Kalypsys, Inc. (US) 2007-08-15 EP disclosed
WO-2006060424-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS KALYPSYS, INC. (US) 2006-06-08 WO disclosed